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GSK-1016790A | TRPV4 channel activator
From $68.00CAS:942206-85-1Catalog Number:10-1198Activity:TRPV4 channel activatorChemical Name:(N-((1S)-1-{[4-((2S)-2-{[(2,4-Dichlorophenyl)sulfonyl]amino}-3-hydroxypropanoyl)-1-piperazinyl]carbonyl}-3-methylbutyl)-1-benzothiophene-2-carboxamideMolecular Weight:655.62Molecular Formula:C28H32Cl2N4O6S2Solubility:Soluble in DMSO (up to 10 mg/ml).Physical Properties:solidPurity:98% by TLC
NMR (Conforms)Storage Temperature:-20°CStability:Stable for 2 years from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 2 months.Shipping Code:RT -
GSK-690693 HCl | Akt inhibitor
From $98.00CAS:937174-76-0Catalog Number:10-1310Activity:Akt inhibitorChemical Name:(S)-4-(2-(4-Amino-1,2,5-oxadiazol-3-yl)-1-ethyl-7-(piperidin-3-ylmethoxy)-1H-imidazo[4,5-c]pyridine-4-yl)-2-methylbut-3-yn-2-ol HClMolecular Weight:461.96Molecular Formula:C21H27N7O3 HClSolubility:Soluble in DMSO (up to 10 mg/ml) or in Ethanol (up to 30 mg/ml).Physical Properties:Off-white solidPurity:99% by HPLC
NMR (Conforms)Storage Temperature:-20°CStability:Stable for 2 years from date of purchase as supplied. Solutions in DMSO or distilled water may be stored at -20° for up to 1 month.Shipping Code:RT -
GSK-J1 | JMJ H3K27 Demethylase inhibitor (Non-cell permeable)
From $75.00CAS:1373422-53-7Catalog Number:10-1393Activity:JMJ H3K27 Demethylase inhibitor (Non-cell permeable)Chemical Name:N-[2-(2-Pyridinyl)-6-(1,2,4,5-tetrahydro-3H-3-benzazepin-3-yl)-4-pyrimidinyl]-β-alanineMolecular Weight:389.46Molecular Formula:C22H23N5O2Solubility:Soluble in DMSO (up to 20 mg/ml).Physical Properties:Pale yellow solidPurity:99% by TLC
NMR (Conforms)Storage Temperature:RTStability:Stable for 2 years from date of purchase as supplied. Solutions in DMSO may be stored at -20° for up to 3 months.Shipping Code:RT