Lipid Receptor Agonists & Antagonists
-
Grapiprant | EP4 Receptor antagonist
From $80.00CAS:415903-37-6Catalog Number:10-4006Activity:EP4 Receptor antagonistChemical Name:1—[2-[4-(2-Ethyl-4,6-dimethylimidazo[4,5-c]pyridine-1-yl)phenyl]ethyl]-3-(4-methylphenyl)sulfonylureaAlternate Names:CJ-023423; ARY-007Molecular Weight:491.61Molecular Formula:C26H29N5O3SSolubility:Soluble in DMSO (up to at least 10 mg/ml)Physical Properties:Off-white solidPurity:98% by TLC
NMR (Conforms)Storage Temperature:-20°CStability:Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 3 months.Shipping Code:RT -
GRI-977143 | LPA2 antagonist
From $80.00CAS:325850-80-5Catalog Number:10-1442Activity:LPA2 antagonistChemical Name:2-[[3-(1,3-dioxo-1H-benz[de]isoquinolin-2(3H)-yl)propyl]thio]benzoic acidMolecular Weight:391.44Molecular Formula:C22H17NO6SSolubility:Soluble in DMSO (up to 35 mg/ml)Physical Properties:White solidPurity:98% by TLC
NMR (Conforms)Storage Temperature:-20°C (des.)Stability:Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 3 months.Shipping Code:RT -
GSK-137647 | GPR120 agonist
From $90.00CAS:349085-82-1Catalog Number:10-1516Activity:GPR120 agonistChemical Name:4-Methoxy-N-(2,4,6-trimethylphenyl)benzenesulfonamideMolecular Weight:305.40+L302Molecular Formula:C16H19NO3SSolubility:Soluble in DMSO (up to 50 mg/ml) or in Ethanol (up to 8 mg/ml with warming).Physical Properties:Off-white solidPurity:98% by TLC
NMR (Conforms)Storage Temperature:-20°CStability:Stable for 2 years from date of purchase as supplied. Solutions in DMSO or ethanol may be stored at -20° for up to 1 month.Shipping Code:RT -
H2L5186303 | LPA2 antagonist
From $60.00CAS:139262-76-3Catalog Number:10-1452Activity:LPA2 antagonistChemical Name:(Z,Z)-4,4′-[1,3-Phenylenebis(oxy-4,1-phenyleneimino)]bis[4-oxo-2-butenoic acid]Molecular Weight:488.45Molecular Formula:C26H202O8Solubility:Soluble in DMSO (up to 50 mg/ml).Physical Properties:Yellow solidPurity:98% by TLC
NMR (Conforms)Storage Temperature:-20°CStability:Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 1 month.Shipping Code:RT
