Epigenetics
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Tenovin-1 | SIRT1/2 inhibitor
From $40.00CAS:380315-80-0Catalog Number:10-2982Activity:SIRT1/2 InhibitorChemical Names:N-[(4-Acetamidophenyl)carbamothioyl]-4-tert-butylbenzamideMolecular Weight:369.48Molecular Formula:C20H23N3O2SSolubility:Soluble in DMSO (10 mg/ml with warming)Physical Properties:White solidPurity:>98% HPLC
NMR (Conforms)Storage Temperature:-20°CStability:Stable for 2 years from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 3 months.Shipping Code:RT -
Trichostatin A | HDAC inhibitor
From $78.00CAS:58880-19-6Catalog Number:10-2110Activity:HDAC inhibitorAlternate Names:TSAChemical Name:(2E,4E,6R)-7-(4-(Dimethylamino)phenyl)-N-hydroxy-4,6-dimethyl-7-oxo-2,4-heptadienamideMolecular Weight:302.38Molecular Formula:C17H22N2O3Solubility:Soluble in DMSO (up to 15 mg/ml), or in Ethanol (up to 3 mg/ml).Physical Properties:Tan solidPurity:99% by HPLC
NMR (Conforms)Storage Temperature:-20°Stability:Stable for 2 years from date of purchase as supplied. Solutions in DMSO or ethanol may be stored at -20° for up to 3 months.Shipping Code:RT -
UNC0379 | Selective SETD8 inhibitor
From $65.00CAS:1620401-82-2Catalog Number:10-4870Activity:Selective SETD8 inhibitorChemical Name:6,7-Dimethoxy-2-(pyrrolidin-1-yl)-N-(5-(pyrrolidin-1-yl)-pentyl)quinazolin-4-amineMolecular Weight:413.56Molecular Formula:C23H35N5O2Solubility:Soluble in DMSO (up to 30 mg/ml)Physical Properties:Tan solidPurity:98% by TLC
NMR (Conforms)Storage Temperature:-20°CStability:Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 1 month.Shipping Code:RT -
UNC1999 | Methyltransferase inhibitor
From $59.00CAS:1431612-23-5Catalog Number:10-4542Activity:Methyltransferase inhibitorChemical Name:N-[(6-Methyl-2-oxo-4-propyl-1H-pyridin-3-yl)methyl]-1-propan-2-yl-6-[6-(4-propan-2-ylpiperazin-1-yl)pyridin-3-yl]indazole-4-carboxamideMolecular Weight:569.74Molecular Formula:C33H43N7O2Solubility:Soluble in DMSO (up to 10 mg/ml).Physical Properties:White solidPurity:98% by HPLC
NMR (Conforms)Storage Temperature:-20°Stability:Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20° for up to 3 months.Shipping Code:RT
EXPLORE OTHER Cancer
- ADC warheads
- Angiogenesis
- Autophagy
- Cancer Cell Metabolism
- Cancer Stem Cells
- Cell Cycle
- Cellular Stress
- Chemotherapeutics
- Cytoskeleton
- DNA Damage/Repair
- Drug resistance
- Gene Regulation/Transcription
- Growth factors
- Immuno-oncology
- Kinases
- Metastasis
- Other Cancer
- p53 & Other Tumor Suppressors
- Programmed cell death
- Stem Cells
- Ubiquitin proteasome
- Wnt/ß-Catenin
