Kinases Archives | Page 27 of 30

SU9516 | pan-specific CDK inhibitor

CAS:

SU9516

Catalog Number:

10-5705

Activity:

pan-specific CDK inhibitor

Chemical Names:

(Z)-1,3-Dihydro-3-(1H-imidazol-4-ylmethylene)-5-methoxy-2H-2-one

Molecular Weight:

241.25

Molecular Formula:

C₁₃H₁₁N₃O₂

Solubility:

Soluble in DMSO (25 mg/ml)

Physical Properties:

Orange solid

Purity:

>98% HPLC
NMR (Conforms)

Storage Temperature:

-20°C

Stability:

Stable for 2 years from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 2 months.

Shipping Code:

RT

From $75.00
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Sunitinib malate | VEGFR, PDGFR kinase inhibitor

CAS:

341031-54-7

Catalog Number:

10-1078

Activity:

VEGFR, PDGFR kinase inhibitor

Alternate Names:

SU-11248

Chemical Name:

N-[2-(Diethylamino)ethyl]-5-[(Z)-(5-fluoro-1,2-dihydro-2-oxo-3H-indol-3-ylidene)methyl]-2,4-dimethyl-1H-pyrrole-3-carboxamide malate

Molecular Weight:

532.57

Molecular Formula:

C₂₂H₂₇FN₄O₄ C₄H₆O₅

Solubility:

Soluble in DMSO (up to 13 mg/ml).

Physical Properties:

Orange solid

Purity:

98% by TLC
NMR (Conforms)

Storage Temperature:

-20°C

Stability:

Stable for 2 years from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 3 months.

Shipping Code:

RT

From $60.00
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THZ1 | Potent and selective CDK7 inhibitor

CAS:

1604810-83-4

Catalog Number:

10-4120

Activity:

Potent and selective CDK7 inhibitor

Chemical Name:

(E)-N-(3-((5-chloro-4-(1H-indol-3-yl)pyrimidin-2-yl)amino)phenyl)-4-(4-(dimethylamino)but-2-enamido)benzamide

Molecular Weight:

566.05

Molecular Formula:

C₃₁H₂₈ClN₇O₂

Solubility:

Soluble in DMSO (up to at least 25 mg/ml)

Physical Properties:

Tan solid

Purity:

97% by TLC
NMR (Conforms)

Storage Temperature:

-20°C

Stability:

Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 3 months.

Shipping Code:

RT

From $80.00
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Torin1 | mTOR inhibitor

CAS:

1222998-36-8

Catalog Number:

10-3013

Activity:

mTOR inhibitor

Chemical Name:

1-[4-[4-(1-Oxopropyl)-1-piperazinyl]-3-(trifluoromethyl)phenyl]-9-(3-quinolinyl)-benzo[h]-1,6-naphthyridin-2(1H)-one

Molecular Weight:

607.62

Molecular Formula:

C₃₅H₂₈F₃N₅O₂

Solubility:

Soluble in DMSO (up to 8 mg/ml).

Physical Properties:

White or off-white solid

Purity:

98% by HPLC
NMR (Conforms)

Storage Temperature:

-20°C

Stability:

Stable for 2 years from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 2 months.

Shipping Code:

RT

From $70.00
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Tozasertib | Aurora kinase inhibitor

CAS:

639089-54-6

Catalog Number:

10-2178

Activity:

Aurora kinase inhibitor

Alternate Names:

VX-680, MK-0457

Molecular Weight:

464.59

Molecular Formula:

C₂₃H₂₈N₈OS

Solubility:

Soluble in DMSO (up to 100 mg/ml).

Physical Properties:

Off-white solid

Purity:

99% by HPLC
NMR (Conforms)

Storage Temperature:

-20°

Stability:

Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20° for up to 3 months.

Shipping Code:

RT

From $50.00
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Kinases

SU9516 | pan-specific CDK inhibitor

Sunitinib malate | VEGFR, PDGFR kinase inhibitor

THZ1 | Potent and selective CDK7 inhibitor

Torin1 | mTOR inhibitor

Tozasertib | Aurora kinase inhibitor

EXPLORE OTHER Cancer

Focus Biomolecules • Plymouth Meeting, PA USA • 1-855-FOCUS21

Focus Biomolecules
Plymouth Meeting, PA USA
1-855-FOCUS21

Kinases

SU9516 | pan-specific CDK inhibitor

Sunitinib malate | VEGFR, PDGFR kinase inhibitor

THZ1 | Potent and selective CDK7 inhibitor

Torin1 | mTOR inhibitor

Tozasertib | Aurora kinase inhibitor

EXPLORE OTHER Cancer

Focus Biomolecules • Plymouth Meeting, PA USA • 1-855-FOCUS21

Focus Biomolecules Plymouth Meeting, PA USA1-855-FOCUS21

Focus Biomolecules
Plymouth Meeting, PA USA
1-855-FOCUS21