Insulin Receptor

  • GSK2656157 | PERK inhibitor

    CAS:
    1337532-29-2
    Catalog Number:
    10-4855
    Activity:
    PERK inhibitor
    Chemical Names:
    1-[5-(4-Amino-7-methylpyrrolo[2,3-d]pyrimidin-5-yl)-4-fluoro-2,3-dihydroindol-1-yl]-2-(6-methylpyridin-2-yl)ethanone
    Molecular Weight:
    416.45
    Molecular Formula:
    C23H21FN6O
    Solubility:
    Soluble in DMSO (10 mg/ml with warming)
    Physical Properties:
    White solid
    Purity:
    >98% HPLC
    NMR (Conforms)
    Storage Temperature:
    -20°C
    Stability:
    Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 1 month.
    Shipping Code:
    RT
    From $40.00
  • GW1100 | GPR40 antagonist

    CAS:
    306974-70-9
    Catalog Number:
    10-4516
    Activity:
    GPR40 antagonist
    Chemical Name:
    1-(4-Ethoxycarbonylphenyl-2-(4-fluorobenzylthio)-5-(2-ethoxy-5-pyrimidinylmethyl)-4-pyrimidinone
    Molecular Weight:
    520.59
    Molecular Formula:
    C27H25FN4O4S
    Solubility:
    Soluble in DMSO (up to 2 mg/ml) or in DMF (up to 5 mg/ml).
    Physical Properties:
    White solid
    Purity:
    96% by LCMS
    NMR (Conforms)
    Storage Temperature:
    -20°
    Stability:
    Stable for 1 year from date of purchase as supplied. Solutions in DMSO or DMF may be stored at -20° for up to 3 months. Dilutions into aqueous media are not stable and should be used within one working day.
    Shipping Code:
    RT
    From $50.00
  • ISX9 | Neurogenic differentiation inducer

    CAS:
    832115-62-5
    Catalog Number:
    10-1357
    Activity:
    Neurogenic differentiation inducer
    Chemical Name:
    N-Cyclopropyl-5-(2-thienyl)-3-isoxazolecarboxamide
    Molecular Weight:
    234.28
    Molecular Formula:
    C11H10N2O2S
    Solubility:
    Soluble in DMSO (up to 60 mg/ml) or in Ethanol (up to 16 mg/ml).
    Physical Properties:
    Tan solid
    Purity:
    99% by TLC
    NMR (Conforms)
    Storage Temperature:
    -20°
    Stability:
    Stable for 2 years from date of purchase as supplied. Solutions in DMSO or ethanol may be stored at -20° for up to 3 months.
    Shipping Code:
    RT
    From $66.00
  • KY-226 | PTP1B inhibitor

    CAS:
    1621673-53-7
    Catalog Number:
    10-4004
    Activity:
    PTP1B Inhibitor
    Chemical Name:
    4-(Biphenyl-4-ylmethylsulfanylmethyl)-N-(hexane-1-sulfonyl)benzoylamide
    Molecular Weight:
    481.67
    Molecular Formula:
    C27H31NO3S2
    Solubility:
    Soluble in DMSO (>25 mg/ml).
    Physical Properties:
    Off-white solid
    Purity:
    >98% by TLC
    NMR (Conforms)
    Storage Temperature:
    -20°
    Stability:
    Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20° for up to 3 months.
    Shipping Code:
    RT
    From $65.00
  • Obeticholic Acid | FXR agonist

    CAS:
    459789-99-2
    Catalog Number:
    10-2838
    Activity:
    FXR agonist
    Chemical Name:
    3α-7α-dihydroxy-6α-ethyl-5ß-cholan-24-oic acid
    Alternate Names:
    6-Ethylchenodeoxycholic acid; 6-ECDCA
    Molecular Weight:
    420.63
    Molecular Formula:
    C26H44O4
    Solubility:
    Soluble in DMSO (up to 35 mg/ml) or in Ethanol (up to 25 mg/ml)
    Physical Properties:
    White solid
    Purity:
    98% by TLC
    NMR (Conforms)
    Storage Temperature:
    -20°C
    Stability:
    Stable for 2 years from date of purchase as supplied. Solutions in DMSO or ethanol may be stored at -20°C for up to 2 months.
    Shipping Code:
    RT
    From $50.00
1 2 3 4 5