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GSK2879552 | Potent and selective LSD1 inhibitor
From $80.00CAS:1401966-69-5Catalog Number:10-4020Activity:Potent and selective LSD1 inhibitorChemical Name:4-[[4-[[[(1R,2S)-2-Phenylcyclopropyl]amino]methyl]-1-piperidinyl]methyl]benzoic acid dihydrochlorideMolecular Weight:437.40Molecular Formula:C23H28N2O2 • HClSolubility:Soluble in DMSO (up to 25 mg/ml) or in Water (up to at least 25 mg/ml)Physical Properties:White solidPurity:98% by HPLC
NMR (Conforms)Storage Temperature:-20°CStability:Stable for 1 year from date of purchase as supplied. Solutions in DMSO or distilled water may be stored at -20°C for up to 3 months.Shipping Code:RT -
GSK2982772 | RIP1 inhibitor
From $95.00CAS:1622848-92-3Catalog Number:10-4792Activity:RIP1 kinase inhibitorChemical Names:(S)-5-Benzyl-N-(5-methyl-4-oxo-2,3,4,5-tetrahydrobenzo[b]-[1,4]oxazepin-3-yl)-4H-1,2,4-traizole-3-carboxamide; GSK772Molecular Weight:377.40Molecular Formula:C20H19N5O3Solubility:Soluble in DMSO (>25 mg/ml)Physical Properties:Off-white solidPurity:>98% HPLC
NMR (Conforms)Storage Temperature:-20°CStability:Stable for 2 year from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 1 month.Shipping Code:RT -
GSK3326595 | Selective PRMT5 inhibitor
From $50.00CAS:1616392-22-3Catalog Number:10-4028Activity:Selective PRMT5 inhibitorChemical Name:6-[(1-Acetylpiperidine-4-yl)amino]-N-[(2S)-3-(3,4-dihydro-1H-isoquinolin-2-yl)-2-hydroxypropyl]pyrimidine-4-carboxamideAlternate Name:EPZ015938Molecular Weight:452.56Molecular Formula:C24H32N6O3Solubility:Soluble in DMSO (up to 20 mg/ml).Physical Properties:Off-white solidPurity:98% by HPLC
NMR (Conforms)Storage Temperature:-20°Stability:Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20° for up to 1 month.Shipping Code:RT -
GSK4112 | Rev-Erbα agonist
From $55.00CAS:1216744-19-2Catalog Number:10-5493Activity:Rev-Erbα agonistChemical Names:N-[(4-Chlorophenyl)methyl]-N-[(5-nitro-2-thienyl)methyl]glycine, 1,1-dimethyl esterAlternate Name:SR6452Molecular Weight:396.89Molecular Formula:C18H21ClN2O4SSolubility:Soluble in DMSO (50 mg/ml)Physical Properties:White solidPurity:>98% HPLC
NMR (Conforms)Storage Temperature:-20°CStability:Stable for 2 years from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 2 months.Shipping Code:RT -
GSK417651A | TRPC3/6 blocker
From $100.00CAS:736945-96-3Catalog Number:10-1434Activity:TRPC3/6 blockerChemical Name:(3,4-Dihydroisoquinolin-2(1H)-yl)(2-((4-methoxyphenyl)amino)thiazol-4-yl)methanoneMolecular Weight:365.46Molecular Formula:C20H19N3O2SSolubility:Soluble in DMSO (up to 50 mg/ml) or in Ethanol (up to 15 mg/ml with warming).Physical Properties:Yellow solidPurity:99% by HPLC
NMR (Conforms)Storage Temperature:RT (des.)Stability:Stable for 1 year from date of purchase as supplied. Solutions in DMSO or ethanol may be stored at -20° for up to 3 months.Shipping Code:RT