Highly Selective Inhibitors
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GSK2334470 | Potent and selective PDK1 inhibitor
From $59.00CAS:1227911-45-6Catalog Number:10-4725Activity:Potent and selective PDK1 inhibitorChemical Name:(3S,6R)-1-[6-(3-Amino-1H-indazol-6-yl)-2-(methylamino)-4-pyrimidinyl]-N-cyclohexyl-6-methyl-3-piperidinecarboxamideMolecular Weight:462.60Molecular Formula:C25H34N8OSolubility:Soluble in DMSO (> 25 mg/ml).Physical Properties:Off-white solidPurity:>98% by HPLC
NMR (Conforms)Storage Temperature:-20° (des.)Stability:Stable for 1 year as supplied. Solutions in DMSO may be stored at -20° for up to 3 months.Shipping Code:RT -
GSK2656157 | PERK inhibitor
From $40.00CAS:1337532-29-2Catalog Number:10-4855Activity:PERK inhibitorChemical Names:1-[5-(4-Amino-7-methylpyrrolo[2,3-d]pyrimidin-5-yl)-4-fluoro-2,3-dihydroindol-1-yl]-2-(6-methylpyridin-2-yl)ethanoneMolecular Weight:416.45Molecular Formula:C23H21FN6OSolubility:Soluble in DMSO (10 mg/ml with warming)Physical Properties:White solidPurity:>98% HPLC
NMR (Conforms)Storage Temperature:-20°CStability:Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 1 month.Shipping Code:RT -
GSK583 | RIP2 kinase inhibitor
From $40.00CAS:1346547-00-9Catalog Number:10-4761Activity:RIP2 kinase inhibitorChemical Name:6-tert-Butylsulfonyl-N-(5-fluoro-1H-indazol-3-yl)quinoline-4-amineMolecular Weight:398.45Molecular Formula:C20H19FN4O2SSolubility:Soluble in DMSO (up to at least 25 mg/ml).Physical Properties:Pale yellow solidPurity:98% by HPLC
NMR (Conforms)Storage Temperature:-20°Stability:Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20° for up to 1 month.Shipping Code:RT
