Other Kinases
-
Larotrectinib | TRK inhibitor
From $60.00CAS:1223403-58-4Catalog Number:10-4832Activity:Potent and selective panTRK inhibitorChemical Name:(3S)-N-[5-[(2R)-2-(2,5-Difluorophenyl)pyrrolidine-1-yl]pyrazolo[1,5-a]pyrimidin-3-yl]-3-hydroxypyrrolidine-1-carboxamideAlternate Name:LOXO-101; ARRY-470Molecular Weight:428.44Molecular Formula:C21H22F2N5O2Solubility:Soluble in DMSO (up to 5 mg/ml).Physical Properties:Yellow solidPurity:98% by HPLC
NMR (Conforms)Storage Temperature:RTStability:Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20° for up to 2 months.Shipping Code:RT -
Lestaurtinib | FLT3/TrkA inhibitor
From $50.00CAS:111358-88-4Catalog Number:10-2149Activity:FLT3/TrkA inhibitorAlternate Names:KT5555; CEP-701Molecular Weight:439.46Molecular Formula:C26H21N3O4Solubility:Soluble in DMSO (up to 100 mg/ml) or in Ethanol (up to 20 mg/ml)Physical Properties:White or off-white solidPurity:98% by TLC
NMR (Conforms)Storage Temperature:-20°C (des.)Stability:Stable for 1 year from date of purchase as supplied. Solutions in DMSO or ethanol may be stored at -20°C for up to 1 month.Shipping Code:RT -
LH-846 | Casein kinase 1 delta inhibitor
From $55.00CAS:639052-78-1Catalog Number:10-1465Activity:Casein kinase 1 delta inhibitorChemical Name:N-(5-Chloro-6-methyl-2-benzothiazolyl)benzeneacetamideMolecular Weight:316.81Molecular Formula:C16H13ClN2OSSolubility:Soluble in DMSO (up to 20 mg/ml) or in Ethanol (up to 5 mg/ml with warming).Physical Properties:White solidPurity:98% by TLC
NMR (Conforms)Storage Temperature:RTStability:Stable for 1 year from date of purchase as supplied. Solutions in DMSO or ethanol may be stored at -20°C for up to 3 months.Shipping Code:RT -
Linsitinib | Inhibits IGF-1R kinase and InsR kinase
From $60.00CAS:867160-71-2Catalog Number:10-4814Activity:Inhibits IGF-1R kinase and InsR kinaseChemical Name:3-[8-Amino-1-(2-phenyl-7-quinolyl)imidazo[1,5-a]pyrazin-3-yl]-1-methyl-cyclobutanolAlternate Names:OSI-906Molecular Weight:421.49Molecular Formula:C26H23N5OSolubility:Soluble in DMSO (up to 30 mg/ml)Physical Properties:Yellow solidPurity:98% by HPLC
NMR (Conforms)Storage Temperature:-20°CStability:Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 2 months.Shipping Code:RT -
Lonidamine | Inhibits Cancer Cell Metabolism
From $45.00CAS:50264-69-2Catalog Number:10-4563Activity:Decreases aerobic and anaerobic glycolysis in tumor cellsAlternate Names:AF1890; Diclondazolic acidChemical Name:1-[(2,4-Dichlorophenyl)methyl]-1H-indazole-3-carboxylic acidMolecular Weight:321.16Molecular Formula:C15H10Cl2N2O2Solubility:Soluble in DMSO (up to 25 mg/ml).Physical Properties:White solidPurity:98% by TLC
NMR (Conforms)Storage Temperature:-20°Stability:Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20° for up to 1 month.Shipping Code:RT
