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Duvelisib | PI3Kdelta/gamma inhibitor
From $65.00CAS:1201438-56-3Catalog Number:10-4788Activity:PI3Kδ/γ inhibitor/Cancer immunotherapy enhancerChemical Name:8-Chloro-2-phenyl-3-[(1S)-1-(7H-purin-6-ylamino)ethyl]isoquinolin-1-oneAlternative Name:IPI-145Molecular Weight:416.87Molecular Formula:C22H17ClN6OSolubility:Soluble in DMSO (up to at least 25 mg/ml)Physical Properties:White solidPurity:98% by HPLC
NMR (Conforms)Storage Temperature:-20°CStability:Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 3 months.Shipping Code:RT -
GDC-0941 | pan-PI3K inhibitor
From $58.00CAS:957054-30-7Catalog Number:10-2141Activity:pan-Class I PI3-kinase inhibitorChemical Names:4-[2-(1H-Indazol-4-yl)-6-[(4-methylsulfonylpiperazin-1-yl)methyl]thieno[3,2-d]pyrimidin-4-yl]morpholine; PictilisibMolecular Weight:513.64Molecular Formula:C23H27N7O3S2Solubility:Soluble in DMSO (>25 mg/ml)Physical Properties:White/off-white solidPurity:99% HPLC
NMR (Conforms)Storage Temperature:-20°CStability:Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 3 months.Shipping Code:RT -
Idelalisib | Selective PI3Kδ Inhibitor
From $60.00CAS:870281-82-6Catalog Number:10-4820Activity:Selective PI3Kδ InhibitorChemical Name:5-Fluoro-3-phenyl-2-[(1S)-1-(7H-purin-6-ylamino)propyl]quinazolin-4-oneAlternate Names:CAL-101Molecular Weight:415.43Molecular Formula:C21H18FN7OSolubility:Soluble in DMSO (>25 mg/ml)Physical Properties:White solidPurity:>98% by HPLC
NMR (Conforms)Storage Temperature:-20°CStability:Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 2 months.Shipping Code:RT -
IPI-549 | Selective PI3Kgamma inhibitor / Immuno-oncology agent
From $50.00CAS:1693758-51-8Catalog Number:10-4827Activity:Selective PI3K-gamma inhibitor / Immuno-oncology agentChemical Name:(S)-2-Amino-N-[1-[8-[2-(1-methylpyrazol-4-yl)ethynyl]-1-oxo-2-phenylisoquinolin-3-yl]ethyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide; EganelisibMolecular Weight:629.68Molecular Formula:C30H24N8O2Solubility:Soluble in DMSO (up to at least 25 mg/ml)Physical Properties:Pale yellow solidPurity:98% by HPLC
NMR (Conforms)Storage Temperature:-20°CStability:Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 1 month.Shipping Code:RT