Proteasome

  • ML241 | p97 AAA ATPase inhibitor

    CAS:
    1346528-06-0
    Catalog Number:
    10-1555
    Activity:
    p97 AAA ATPase inhibitor
    Chemical Name:
    N-Benzyl-2-(2,3-dihydro-1,4-benzoxazin-4-yl)-5,6,7,8-tetrahydroquinazolin-4-amine
    Alternate Name:
    CID49830260
    Molecular Weight:
    372.46
    Molecular Formula:
    C23H24N4O
    Solubility:
    Soluble in DMSO (up to 50 mg/ml) or in Ethanol (up to 14 mg/ml with warming).
    Physical Properties:
    Pale yellow solid
    Purity:
    98% by HPLC
    NMR (Conforms)
    Storage Temperature:
    -20°
    Stability:
    Stable for 1 year from date of purchase as supplied. Solutions in DMSO or ethanol may be stored at -20° for up to 3 months.
    Shipping Code:
    RT
    From $90.00
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  • MLN4924 | NEDD8 activating enzyme inhibitor

    CAS:
    905579-51-3
    Catalog Number:
    10-1311
    Activity:
    NEDD8 activating enzyme inhibitor
    Chemical Name:
    ((1S,2S,4R)-4-(4-(((S)-2,3-Dihydro-1H-inden-1-yl)amino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2-hydroxycyclopentyl)methyl sulfamate; Pevonedistat
    Molecular Weight:
    443.53
    Molecular Formula:
    C21H25N5O4S
    Solubility:
    Soluble in DMSO (up to 10 mg/ml).
    Physical Properties:
    White solid
    Purity:
    98% by TLC
    NMR (Conforms)
    Storage Temperature:
    -20°C (des.)
    Stability:
    Stable for 2 years from date of purchase as supplied. Solutions in DMSO may be stored at -20° for up to 3 months.
    Shipping Code:
    RT
    From $60.00
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  • Pyr41 | E1 UAE inhibitor

    CAS:
    418805-02-4
    Catalog Number:
    10-1304
    Activity:
    E1 UAE inhibitor
    Chemical Name:
    4-[4-(5-Nitro-furan-2-ylmethylene)-3,5-dioxo-pyrazolidin-1-yl]-benzoic acid ethyl ester
    Molecular Weight:
    371.31
    Molecular Formula:
    C17H13N3O7
    Solubility:
    Soluble in DMSO (up to 25 mg/ml).
    Physical Properties:
    Brown solid
    Purity:
    98% by TLC
    NMR (Conforms)
    Storage Temperature:
    -20°C (des.)
    Stability:
    Stable for 2 years from date of purchase as supplied. Solutions in DMSO may be stored at -20° for up to 1 week.
    Shipping Code:
    RT
    From $55.00
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  • Suc-Leu-Leu-Val-Tyr-AMC | Proteasome substrate

    CAS:
    94367-21-2
    Catalog Number:
    10-2971
    Activity:
    Proteasome substrate
    Alternate Names:
    Suc-LLVY-AMC, Proteasome Substrate III (Fluorogenic)
    Molecular Weight:
    763.88
    Molecular Formula:
    C40H53N5O10
    Solubility:
    Soluble in DMSO (up to 20 mg/ml), or in DMF (up to 10 mg/ml)
    Physical Properties:
    Lyophilized solid
    Purity:
    98% by HPLC
    NMR (Conforms)
    Storage Temperature:
    -20°C
    Stability:
    Stable for 1 year from date of purchase as supplied. Solutions in DMSO or DMF may be stored at -20°C for up to 1 month.
    Shipping Code:
    RT
    From $30.00
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  • Z-Leu-Leu-Leu-vinylsulfone | Proteasome inhibitor

    CAS:
    193482-47-2
    Catalog Number:
    10-4990
    View Product This product has multiple variants. The options may be chosen on the product page
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