Chemotherapeutics
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Lapatinib (base) | EGFR and HER2 inhibitor
From $55.00CAS:231277-92-2Catalog Number:10-2147Activity:EGFR and HER2 inhibitorChemical Name:N-[3-Chloro-4-[(3-fluorophenyl)methoxy]phenyl]-6-[5-[(2-methylsulfonylethylamino)methyl]-2-furyl]quinazolin-4-amineAlternate Names:GW-572016Molecular Weight:581.06Molecular Formula:C29H26ClFN4O4SSolubility:Soluble in DMSO (up to 200 mg/ml)Physical Properties:Yellow solidPurity:98% by TLC
NMR (Conforms)Storage Temperature:-20°CStability:Stable for 2 years from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 1 month.Shipping Code:RT -
Larotrectinib | TRK inhibitor
From $60.00CAS:1223403-58-4Catalog Number:10-4832Activity:Potent and selective panTRK inhibitorChemical Name:(3S)-N-[5-[(2R)-2-(2,5-Difluorophenyl)pyrrolidine-1-yl]pyrazolo[1,5-a]pyrimidin-3-yl]-3-hydroxypyrrolidine-1-carboxamideAlternate Name:LOXO-101; ARRY-470Molecular Weight:428.44Molecular Formula:C21H22F2N5O2Solubility:Soluble in DMSO (up to 5 mg/ml).Physical Properties:Yellow solidPurity:98% by HPLC
NMR (Conforms)Storage Temperature:RTStability:Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20° for up to 2 months.Shipping Code:RT -
Lenalidomide | Immunomodulator
From $75.00CAS:191732-72-6Catalog Number:10-2148Activity:ImmunomodulatorChemical Name:(R,S)-3-(4-Amino-1-oxo-3H-isoindol-2-yl)piperidine-2,6-dioneMolecular Weight:259.26Molecular Formula:C13H13N3O3Solubility:Soluble in DMSO (up to 30 mg/ml)Physical Properties:White solidPurity:98% by TLC
NMR (Conforms)Storage Temperature:RTStability:Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 3 months.Shipping Code:RT -
Lenvatinib | VEGFR inhibitor
From $55.00CAS:417716-92-8Catalog Number:10-3313Activity:VEGFR inhibitorChemical Name:4-[3-Chloro-4-[[(cyclopropylamino)carbonyl]amino]phenoxy]-7-methoxy-6-quinolinecarboxamideAlternate Names:E7080Molecular Weight:426.85Molecular Formula:C21H19ClN4O4Solubility:Soluble in DMSO (up to 20 mg/ml)Physical Properties:White solidPurity:98% by HPLC
NMR (Conforms)Storage Temperature:-20°CStability:Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 3 months.Shipping Code:RT -
Methotrexate | Dihydrofolate reductase inhibitor
From $50.00CAS:133073-73-1Catalog Number:10-1260Activity:Dihydrofolate reductase inhibitorChemical Names:N-[4-[[(2,4-Diamino-6-pteridinyl)methyl]methylamino]benzoyl]-L-glutamic acid; Amethopterin; CL-14377; NSC740Molecular Weight:683.63Molecular Formula:C20H22N8O5·XH2OSolubility:Soluble in DMSO (45 mg/ml)Physical Properties:Yellow solidPurity:>98% HPLC
NMR (Conforms)Storage Temperature:-20°CStability:Stable for 2 years from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 3 months.Shipping Code:RT
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