Kinases Archives

Vandetanib | VEGFR2 inhibitor

CAS:

443913-73-3

Catalog Number:

10-2185

Activity:

VEGFR2 inhibitor

Chemical Names:

4-(4-Bromo-2-fluoroanilino)-6-methoxy-7-(1-methylpiperidin-4-yl)methoxy]quinazoline

Alternate Name:

ZD6474

Molecular Weight:

475.35

Molecular Formula:

C₂₂H₂₄BrFN₄O₂

Solubility:

Soluble in DMSO (30 mg/ml); Ethanol (10 mg/ml with warming)

Physical Properties:

White to off-white solid

Purity:

98% TLC
NMR (Conforms)

Storage Temperature:

-20°C

Stability:

Stable for 2 years from date of purchase as supplied. Solutions in DMSO or ethanol may be stored at -20°C for up to 1 month.

Shipping Code:

RT

From $50.00
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Vatalanib 2HCl | VEGFR kinase inhibitor

CAS:

212141-51-0

Catalog Number:

10-2183

Activity:

VEGFRK inhibitor

Chemical Name:

N-(4-Chlorophenyl)-4-(4-pyridinylmethyl)-1-phthalazinamine dihydrochloride

Alternate Names:

CGP-79787; PTK-787; ZK222584

Molecular Weight:

419.73

Molecular Formula:

C₂₀H₁₅ClN₄·2HCl

Solubility:

Soluble in DMSO (up to 20 mg/ml with warming) or in Water (up to 100 mg/ml)

Physical Properties:

White or off-white solid

Purity:

98% by TLC
NMR (Conforms)

Storage Temperature:

-20°C

Stability:

Stable for 2 years from date of purchase as supplied. Solutions in DMSO or distilled water may be stored at -20°C for up to 3 months.

Shipping Code:

RT

From $50.00
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VE-821 | Potent and selective ATR inhibitor

CAS:

1232410-49-9

Catalog Number:

10-5589

Activity:

ATR inhibitor

Chemical Names:

3-Amino-6-[4-(methlsulfonyl)phenyl)-N-phenyl-2-pyrazinecarboxamide

Molecular Weight:

368.41

Molecular Formula:

C₁₈H₁₆N₄O₃S

Solubility:

Soluble in DMSO (40 mg/ml)

Physical Properties:

Beige solid

Purity:

>98% HPLC
NMR (Conforms)

Storage Temperature:

-20°C

Stability:

Stable for 2 years from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 1 month.

Shipping Code:

RT

From $80.00
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Volasertib | Potent and selective inhibitor of Polo-like kinase 1

CAS:

755038-65-4

Catalog Number:

10-4818

Activity:

Potent and selective inhibitor of Polo-like kinase 1

Chemical Name:

N-[4-[4-(Cyclopropylmethyl)piperazin-1-yl]cyclohexyl]-4-[[(7R)-7-ethyl-5-methyl-6-oxo-8-propan-2-yl-7H-pteridin-2-yl]amino]-3-methoxybenzamide

Alternate Name:

BI 6727

Molecular Weight:

618.82

Molecular Formula:

C₃₄H₅₀N₈O₃

Solubility:

Soluble in DMSO (up to at least 25 mg/ml).

Physical Properties:

Off-white solid

Purity:

98% by HPLC
NMR (Conforms)

Storage Temperature:

-20°

Stability:

Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20° for up to 1 month.

Shipping Code:

RT

From $70.00
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WHI-P131 | JAK3 inhibitor

CAS:

202475-60-3

Catalog Number:

10-1190

Activity:

JAK3 inhibitor

Alternate Names:

JANEX-1

Chemical Name:

4-[(4′-Hydroxyphenyl)amino]-6,7-dimethoxyquinazoline

Molecular Weight:

333.78

Molecular Formula:

C₁₆H₁₅N₃O₃·HCl

Solubility:

Soluble in DMSO (up to 50 mg/ml).

Physical Properties:

Yellow solid

Purity:

98% by TLC
NMR (Conforms)

Storage Temperature:

-20°C

Stability:

Stable for 2 years from date of purchase as supplied. Protect from moisture. Solutions in DMSO may be stored at -20°C for up to 2 months.

Shipping Code:

RT

From $60.00
View Product This product has multiple variants. The options may be chosen on the product page

Kinases

Vandetanib | VEGFR2 inhibitor

Vatalanib 2HCl | VEGFR kinase inhibitor

VE-821 | Potent and selective ATR inhibitor

Volasertib | Potent and selective inhibitor of Polo-like kinase 1

WHI-P131 | JAK3 inhibitor

EXPLORE OTHER Cancer

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Plymouth Meeting, PA USA
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Kinases

Vandetanib | VEGFR2 inhibitor

Vatalanib 2HCl | VEGFR kinase inhibitor

VE-821 | Potent and selective ATR inhibitor

Volasertib | Potent and selective inhibitor of Polo-like kinase 1

WHI-P131 | JAK3 inhibitor

EXPLORE OTHER Cancer

Focus Biomolecules • Plymouth Meeting, PA USA • 1-855-FOCUS21

Focus Biomolecules Plymouth Meeting, PA USA1-855-FOCUS21

Focus Biomolecules
Plymouth Meeting, PA USA
1-855-FOCUS21