Highly Selective Inhibitors
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MK-2206 | Potent and selective AKT inhibitor
From $60.00CAS:1032350-13-2Catalog Number:10-4801Activity:Potent and selective AKT inhibitorChemical Name:8-(4-(1-Aminocyclobutyl)phenyl-9-phenyl-2H-[1,2,4]triazolo[3,4-f][1,6]naphthyridin-3-one dihydrochlorideMolecular Weight:480.39Molecular Formula:C25H21N5O • 2HClSolubility:Soluble in DMSO (up to 10 mg/ml with warming)Physical Properties:Yellow solidPurity:98% by HPLC
NMR (Conforms)Storage Temperature:-20°CStability:Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 3 months.Shipping Code:RT -
ML167 | Clk4 inhibitor
From $75.00CAS:1285702-20-6Catalog Number:10-4543Activity:Clk4 inhibitorChemical Name:[5-[4-[(5-Methylfuran-2-yl)methylamino]quinazolin-6-yl]furan-2-yl]methanolMolecular Weight:335.36Molecular Formula:C19H17N2O3Solubility:Soluble in DMSO (greater than 25 mg/ml).Physical Properties:White solidPurity:>98% by HPLC
NMR (Conforms)Storage Temperature:-20°CStability:Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20° for up to 3 months.Shipping Code:RT -
Necrostatin-34 | RIP1 kinase inhibitor
CAS:375835-43-1Catalog Number:10-4684 -
NU7441 | DNA-PK inhibitor
From $50.00CAS:503468-95-9Catalog Number:10-4810Activity:DNA-PK inhibitorChemical Name:8-Dibenzothiophen-4-yl-2-morpholin-4-ylchromen-4-oneAlternate Name:Ku-57788Molecular Weight:413.49Molecular Formula:C25H19NO3SSolubility:Soluble in DMSO (up to 10 mg/ml with warming).Physical Properties:Off-white to beige solidPurity:98% by TLC
NMR (Conforms)Storage Temperature:-20°Stability:Stable for 1 year as supplied. Solutions in DMSO may be stored at -20° for up to 3 months.Shipping Code:RT -
NVP-BGJ398 | Pan-specific FGFR inhibitor
From $65.00CAS:872511-34-7Catalog Number:10-4817Activity:Pan-specific FGFR inhibitorChemical Name:3-(2,6-Dichloro-3,5-dimethoxyphenyl)-1-(6-{[4-(4-ethyl-1-piperazinyl)phenyl]amino}-4-pyrimidinyl)-1-methylureaAlternate Names:InfigratinibMolecular Weight:560.48Molecular Formula:C26H31Cl2N7O3Solubility:Soluble in DMSO (up to 5 mg/ml)Physical Properties:White solidPurity:98% by HPLC
NMR (Conforms)Storage Temperature:-20°CStability:Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 2 months.Shipping Code:RT
