Sigma receptor

Agonists

PB28 dihydrochloride | Potent sigma2 agonist

CAS:

172907-03-8

Catalog Number:

10-4665

Activity:

High affinity sigma2 ligand

Chemical Names:

1-Cyclohexyl-4-[3-(1,2,3,4-tetrahydro-5-methoxy-1-naphthalenyl)propyl]piperazine dihydrochloride

Molecular Weight:

443.50

Molecular Formula:

C₂₄H₃₈N₂O

Solubility:

Soluble in DMSO (>25 mg/ml) or water (5 mg/ml)

Physical Properties:

White to off-white solid

Purity:

99% HPLC
NMR (Conforms)

Storage Temperature:

-20°C

Stability:

Stable for 1 year as supplied. Solutions in DMSO may be stored at -20°C for up to 2 months.

Shipping Code:

SA4503 | Potent and selective sigma-1 agonist

CAS:

165377-44-6

Catalog Number:

10-4219

Activity:

Potent and selective sigma-1 agonist

Chemical Name:

1-(3,4-Dimethoxyphenethyl)-4-(3-phenylpropyl)piperazine dihydrochloride

Alternate Name:

Cutamesine

Molecular Weight:

441.43

Molecular Formula:

C₂₃H₃₂N₂O₂ • 2HCl

Solubility:

Soluble in DMSO (up to 5 mg/ml) or in Water (up to at least 25 mg/ml)..

Physical Properties:

White solid

Purity:

98% by TLC
NMR (Conforms)

Storage Temperature:

-20° (des.)

Stability:

Stable for 1 year from date of purchase as supplied. Solutions in DMSO or distilled water may be stored at -20° for up to 1 month.

Shipping Code:

Pridopidine | Sigma-1 ligand Neuroprotectant/Neurorestorative

CAS:

346688-38-8

Catalog Number:

10-4003

Activity:

Sigma-1 ligand Neuroprotectant Neurorestorative

Chemical Name:

4-(3-(Methylsulfonyl)phenyl)-1-propylpiperidine

Alternate Name:

ACR16

Molecular Weight:

281.41

Molecular Formula:

C₁₅H₂₃NO₂S

Solubility:

Soluble in DMSO (up to 10 mg/ml).

Physical Properties:

White solid

Purity:

>98% by TLC
NMR (Conforms)

Storage Temperature:

-20°

Stability:

Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20° for up to 3 months.

Shipping Code:

Antagonists

BD1047 dihydrobromide | Selective sigma-1 antagonist

CAS:

138356-21-5

Catalog Number:

10-4210

Activity:

Selective sigma-1 antagonist

Chemical Name:

N-[2-(3,4Dichlorophenyl)ethyl]-N-methyl-2-(dimethylamino)ethylamine dihydrobromide

Molecular Weight:

437.04

Molecular Formula:

C₁₃H₂₀Cl₂N₂ • 2HBr

Solubility:

Soluble in DMSO (up to 20 mg/ml) or in Water (up to 20 mg/ml)

Physical Properties:

Off-white solid

Purity:

98% by HPLC
NMR (Conforms)

Storage Temperature:

-20°C

Stability:

Stable for 1 year from date of purchase as supplied. Solutions in DMSO or distilled water may be stored at -20°C for up to 3 months.

Shipping Code:

BD1063 dihydrochloride | Selective sigma-1 antagonist

CAS:

206996-13-6

Catalog Number:

10-4211

Activity:

Selective sigma-1 antagonist

Chemical Name:

1-[2-(3,4-Dichlorophenyl)ethyl]-4-methylpiperazine dihydrochloride

Molecular Weight:

346.13

Molecular Formula:

C₁₃H₁₈Cl₂N₂ • 2HCl

Solubility:

Soluble in Water (up to at least 25 mg/ml)

Physical Properties:

Off-white solid

Purity:

98% by HPLC
NMR (Conforms)

Storage Temperature:

-20°C

Stability:

Stable for 1 year from date of purchase as supplied. Solutions in distilled water may be stored at -20°C for up to 3 months.

Shipping Code:

NE-100 | Selective sigma-1 antagonist

CAS:

149409-57-4

Catalog Number:

10-4200

Activity:

Selective sigma-1 antagonist

Chemical Name:

4-Methoxy-3-(2-phenylethoxy)-N,N,dipropylbenzeneethanamine hydrochloride

Molecular Weight:

391.97

Molecular Formula:

C₂₃H₃₃NO₂ • HCl

Solubility:

Soluble in DMSO (up to at least 25 mg/ml) or in Water (up to 10 mg/ml)

Physical Properties:

White solid

Purity:

98% by HPLC
NMR (Conforms)

Storage Temperature:

-20°C

Stability:

Stable for 1 year from date of purchase as supplied. Solutions in DMSO or distilled water may be stored at -20°C for up to 3 months.

Shipping Code:

Sigma receptor

Agonists

PB28 dihydrochloride | Potent sigma2 agonist

SA4503 | Potent and selective sigma-1 agonist

Pridopidine | Sigma-1 ligand Neuroprotectant/Neurorestorative

Antagonists

BD1047 dihydrobromide | Selective sigma-1 antagonist

BD1063 dihydrochloride | Selective sigma-1 antagonist

NE-100 | Selective sigma-1 antagonist

Focus Biomolecules • Plymouth Meeting, PA USA • 1-855-FOCUS21

Focus Biomolecules
Plymouth Meeting, PA USA
1-855-FOCUS21

Sigma receptor

Agonists

PB28 dihydrochloride | Potent sigma2 agonist

SA4503 | Potent and selective sigma-1 agonist

Pridopidine | Sigma-1 ligand Neuroprotectant/Neurorestorative

Antagonists

BD1047 dihydrobromide | Selective sigma-1 antagonist

BD1063 dihydrochloride | Selective sigma-1 antagonist

NE-100 | Selective sigma-1 antagonist

Focus Biomolecules • Plymouth Meeting, PA USA • 1-855-FOCUS21

Focus Biomolecules Plymouth Meeting, PA USA1-855-FOCUS21

Focus Biomolecules
Plymouth Meeting, PA USA
1-855-FOCUS21