Kinases Archives

GDC-0941 | pan-PI3K inhibitor

CAS:

957054-30-7

Catalog Number:

10-2141

Activity:

pan-Class I PI3-kinase inhibitor

Chemical Names:

4-[2-(1H-Indazol-4-yl)-6-[(4-methylsulfonylpiperazin-1-yl)methyl]thieno[3,2-d]pyrimidin-4-yl]morpholine; Pictilisib

Molecular Weight:

513.64

Molecular Formula:

C₂₃H₂₇N₇O₃S₂

Solubility:

Soluble in DMSO (>25 mg/ml)

Physical Properties:

White/off-white solid

Purity:

99% HPLC
NMR (Conforms)

Storage Temperature:

-20°C

Stability:

Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 3 months.

Shipping Code:

RT

From $58.00
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Gefitinib | EGFR kinase inhibitor

CAS:

184475-35-2

Catalog Number:

10-1148

Activity:

EGFR-Kinase inhibitor

Alternate Names:

ZD1839, Iressa

Chemical Name:

N-(3-Chloro-4-fluorophenyl)-7-methoxy-6-(3-morpholinopropoxy)quinazolin-4-amine

Molecular Weight:

446.91

Molecular Formula:

C₂₂H₂₄ClFN₄O₃

Solubility:

Soluble in DMSO (up to 40 mg/ml) or in Ethanol (up to 4 mg/ml).

Physical Properties:

Tan solid

Purity:

98% by TLC
NMR (Conforms)

Storage Temperature:

RT

Stability:

Stable for 2 years from date of purchase as supplied. Solutions in DMSO or ethanol may be stored at -20°C for up to 1 month.

Shipping Code:

RT

From $30.00
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Genistein | Genistin aglycone

CAS:

446-72-0

Catalog Number:

10-2139

Activity:

Tyrosine kinase inhibitor

Chemical Name:

5,7-Dihydroxy-3-(4-hydroxyphenyl)-4H-1-benzopyran-4-one

Alternate Names:

4’,5,7-Trihydroxyisoflavone

Molecular Weight:

270.24

Molecular Formula:

C₁₅H₁₀O₅

Solubility:

Soluble in DMSO (up to 25 mg/ml) or in Ethanol (up to 4 mg/ml)

Physical Properties:

Yellow solid

Purity:

98% by TLC
NMR (Conforms)

Storage Temperature:

-20°C

Stability:

Stable for 1 year from date of purchase as supplied. Solutions in DMSO or ethanol may be stored at -20°C for up to 1 week.

Shipping Code:

RT

From $30.00
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Gilteritinib | FLT3 Inhibitor

CAS:

1254053-43-4

Catalog Number:

10-4170

Activity:

FLT3 inhibitor

Chemical Names:

6-Ethyl-3-[3-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]anilino]-5-(oxan-4-ylamino)pyrazine-2-carboxamide; ASP2215

Molecular Weight:

552.72

Molecular Formula:

C₂₉H₄₄N₈O₃

Solubility:

Soluble in DMSO (25 mg/ml)

Physical Properties:

Off-white to pale pink solid

Purity:

>98% HPLC
NMR (Conforms)

Storage Temperature:

-20°C

Stability:

Stable for 1 year as supplied. Solutions in DMSO may be stored at -20°C for up to 3 months.

Shipping Code:

RT

From $45.00
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Glumetinib | Highly selective c-Met inhibitor

CAS:

1642581-63-2

Catalog Number:

10-4690

Activity:

Highly selective c-Met inhibitor

Chemical Names:

6-(1-Methylpyrazol-4-yl)-1-[6-(1-methylpyrazol-4-yl)imidazo[1,2-a]pyridine-3-yl]sulfonylpyrazolo[4,3-b]pyridine: SCC244

Molecular Weight:

459.48

Molecular Formula:

C₂₁H₁₇N₉O₂S

Solubility:

Soluble in DMSO (>25 mg/ml)

Physical Properties:

Beige solid

Purity:

>98% HPLC
NMR (Conforms)

Storage Temperature:

-20°C

Stability:

Stable for 1 year as supplied. Solutions in DMSO may be stored at -20°C for up to 1 month.

Shipping Code:

RT

From $90.00
View Product This product has multiple variants. The options may be chosen on the product page

Kinases

GDC-0941 | pan-PI3K inhibitor

Gefitinib | EGFR kinase inhibitor

Genistein | Genistin aglycone

Gilteritinib | FLT3 Inhibitor

Glumetinib | Highly selective c-Met inhibitor

EXPLORE OTHER Cancer

Focus Biomolecules • Plymouth Meeting, PA USA • 1-855-FOCUS21

Focus Biomolecules
Plymouth Meeting, PA USA
1-855-FOCUS21

Kinases

GDC-0941 | pan-PI3K inhibitor

Gefitinib | EGFR kinase inhibitor

Genistein | Genistin aglycone

Gilteritinib | FLT3 Inhibitor

Glumetinib | Highly selective c-Met inhibitor

EXPLORE OTHER Cancer

Focus Biomolecules • Plymouth Meeting, PA USA • 1-855-FOCUS21

Focus Biomolecules Plymouth Meeting, PA USA1-855-FOCUS21

Focus Biomolecules
Plymouth Meeting, PA USA
1-855-FOCUS21