Kinases
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Ki8751 | VEGFR2 inhibitor
From $39.00CAS:228559-41-9Catalog Number:10-4388Activity:VEGFR2 inhibitorChemical Names:N-(2,4-Difluorophenyl)-N’-[4-[(6,7-dimethoxy-4-quinolinyl)oxy]-2-fluorophenyl]ureaMolecular Weight:469.42Molecular Formula:C24H18F3N3O4Solubility:Soluble in DMSO (15 mg/ml)Physical Properties:White solidPurity:>98% HPLC
NMR (Conforms)Storage Temperature:-20°CStability:Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 3 months.Shipping Code:RT -
KU-55933 | ATM Kinase Inhibitor
From $65.00CAS:587871-26-9Catalog Number:10-1518Activity:ATM Kinase InhibitorChemical Name:2-(4-Morpholinyl)-6-(1-thianthrenyl)-4H-pyran-4-oneMolecular Weight:395.5Molecular Formula:C21H17NO3S2Solubility:Soluble in DMSO (up to 40 mg/ml) or in Ethanol (up to 20 mg/ml)Physical Properties:Tan solidPurity:98% by TLC
NMR (Conforms)Storage Temperature:-20°Stability:Stable for 2 years from date of purchase as supplied. Solutions in DMSO or ethanol may be stored at -20° for up to 1 month.Shipping Code:RT -
KW-2449 | Multikinase inhibitor
From $35.00CAS:1000669-72-6Catalog Number:10-4448Activity:Multikinsae inhibitorChemical Names:[4-[(E)-2-(1H-Indazol-3-yl)ethenyl]phenyl]-(1-piperazinyl)methanoneMolecular Weight:332.40Molecular Formula:C20H20N4OSolubility:Soluble in DMSO (>25 mg/ml)Physical Properties:Pale yellow solidPurity:>97% HPLC
NMR (Conforms)Storage Temperature:-20°CStability:Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 1 month.Shipping Code:RT -
Lapatinib (base) | EGFR and HER2 inhibitor
From $55.00CAS:231277-92-2Catalog Number:10-2147Activity:EGFR and HER2 inhibitorChemical Name:N-[3-Chloro-4-[(3-fluorophenyl)methoxy]phenyl]-6-[5-[(2-methylsulfonylethylamino)methyl]-2-furyl]quinazolin-4-amineAlternate Names:GW-572016Molecular Weight:581.06Molecular Formula:C29H26ClFN4O4SSolubility:Soluble in DMSO (up to 200 mg/ml)Physical Properties:Yellow solidPurity:98% by TLC
NMR (Conforms)Storage Temperature:-20°CStability:Stable for 2 years from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 1 month.Shipping Code:RT -
Larotrectinib | TRK inhibitor
From $60.00CAS:1223403-58-4Catalog Number:10-4832Activity:Potent and selective panTRK inhibitorChemical Name:(3S)-N-[5-[(2R)-2-(2,5-Difluorophenyl)pyrrolidine-1-yl]pyrazolo[1,5-a]pyrimidin-3-yl]-3-hydroxypyrrolidine-1-carboxamideAlternate Name:LOXO-101; ARRY-470Molecular Weight:428.44Molecular Formula:C21H22F2N5O2Solubility:Soluble in DMSO (up to 5 mg/ml).Physical Properties:Yellow solidPurity:98% by HPLC
NMR (Conforms)Storage Temperature:RTStability:Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20° for up to 2 months.Shipping Code:RT
EXPLORE OTHER Cancer
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- Other Cancer
- p53 & Other Tumor Suppressors
- Programmed cell death
- Stem Cells
- Ubiquitin proteasome
