Kinases
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LDN-192960 2HCl | Haspin and DYRK2/3 inhibitor
From $55.00CAS:184582-62-5Catalog Number:10-4836Activity:Haspin and DYRJ2/3 inhibitorChemical Names:3-(2,7-Dimethoxyacridin-9-yl)sulfanylpropan-1-amine dihydrochlorideMolecular Weight:401.35Molecular Formula:C18H20N2O2S·2HClSolubility:Soluble in DMSO (>25 mg/ml); Water (2 mg/ml)Physical Properties:Yellow solidPurity:>98% HPLC
NMR (Conforms)Storage Temperature:-20°CStability:Stable for 1 year from date of purchase as supplied. Solutions in DMSO or water may be stored at -20°C for up to 1 month.Shipping Code:RT -
Lenvatinib | VEGFR inhibitor
From $55.00CAS:417716-92-8Catalog Number:10-3313Activity:VEGFR inhibitorChemical Name:4-[3-Chloro-4-[[(cyclopropylamino)carbonyl]amino]phenoxy]-7-methoxy-6-quinolinecarboxamideAlternate Names:E7080Molecular Weight:426.85Molecular Formula:C21H19ClN4O4Solubility:Soluble in DMSO (up to 20 mg/ml)Physical Properties:White solidPurity:98% by HPLC
NMR (Conforms)Storage Temperature:-20°CStability:Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 3 months.Shipping Code:RT -
Lestaurtinib | FLT3/TrkA inhibitor
From $50.00CAS:111358-88-4Catalog Number:10-2149Activity:FLT3/TrkA inhibitorAlternate Names:KT5555; CEP-701Molecular Weight:439.46Molecular Formula:C26H21N3O4Solubility:Soluble in DMSO (up to 100 mg/ml) or in Ethanol (up to 20 mg/ml)Physical Properties:White or off-white solidPurity:98% by TLC
NMR (Conforms)Storage Temperature:-20°C (des.)Stability:Stable for 1 year from date of purchase as supplied. Solutions in DMSO or ethanol may be stored at -20°C for up to 1 month.Shipping Code:RT -
LFM-A13 | BTK inhibitor
From $55.00CAS:244240-24-2Catalog Number:10-1032Activity:BTK inhibitorChemical Name:(2Z)-2-Cyano-N-(2,5-dibromophenyl)-3-hydroxy-2-butenamideMolecular Weight:360Molecular Formula:C11H8Br2N2O2Solubility:Soluble in DMSO (up to 15 mg/ml) or in Ethanol (up to 15 mg/ml).Physical Properties:White solidPurity:98% by TLC
NMR (Conforms)Storage Temperature:-20°CStability:Stable for 2 years from date of purchase as supplied. PROTECT FROM MOISTURE. Solutions in DMSO or ethanol may be stored at -20°C for up to 3 months.Shipping Code:RT -
Linsitinib | Inhibits IGF-1R kinase and InsR kinase
From $60.00CAS:867160-71-2Catalog Number:10-4814Activity:Inhibits IGF-1R kinase and InsR kinaseChemical Name:3-[8-Amino-1-(2-phenyl-7-quinolyl)imidazo[1,5-a]pyrazin-3-yl]-1-methyl-cyclobutanolAlternate Names:OSI-906Molecular Weight:421.49Molecular Formula:C26H23N5OSolubility:Soluble in DMSO (up to 30 mg/ml)Physical Properties:Yellow solidPurity:98% by HPLC
NMR (Conforms)Storage Temperature:-20°CStability:Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 2 months.Shipping Code:RT
EXPLORE OTHER Cancer
- ADC warheads
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- Cancer Cell Metabolism
- Cancer Stem Cells
- Cell Cycle
- Cellular Stress
- Chemotherapeutics
- Cytoskeleton
- DNA Damage/Repair
- Drug resistance
- Epigenetics
- Gene Regulation/Transcription
- Growth factors
- Immuno-oncology
- Metastasis
- Other Cancer
- p53 & Other Tumor Suppressors
- Programmed cell death
- Stem Cells
- Ubiquitin proteasome
- Wnt/ß-Catenin
