Kinases
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CID-2011756 | PKD inhibitor
From $60.00CAS:638156-11-3Catalog Number:10-1420Activity:PKD inhibitorChemical Name:5-(3-Chlorophenyl)-N-[4-(4-morpholinylmethyl)phenyl]-2-furancarboxamideMolecular Weight:396.88Molecular Formula:C22H21ClN2O3Solubility:Soluble in DMSO (up to 50 mg/ml) or in Ethanol (up to 8 mg/ml with warming).Physical Properties:Tan solidPurity:98% by TLC
NMR (Conforms)Storage Temperature:RTStability:Stable for 1 year from date of purchase as supplied. Solutions in DMSO or ethanol may be stored at -20° for up to 3 months.Shipping Code:RT -
Crenolanib | PDGFR and FLT3 inhibitor
From $60.00CAS:670220-88-9Catalog Number:10-4782Activity:PDGFR and FLT3 inhibitorChemical Name:1-[2-[5-[(3-Methyloxetan-3-yl)methoxy]benzimidazole-1-yl]quinoline-8-yl]piperidin-4-amineAlternate Name:CP-868,596Molecular Weight:443.55Molecular Formula:C26H29N5O2Solubility:Soluble in DMSO (up to 15 mg/ml) or in Ethanol (up to 10 mg/ml).Physical Properties:White solidPurity:>97% by HPLC
NMR (Conforms)Storage Temperature:-20°Stability:Stable for 1 year as supplied. Solutions in DMSO or ethanol may be stored at -20° for up to 1 month.Shipping Code:RT -
Crizotinib | c-MET and ALK inhibitor
From $80.00CAS:877399-52-5Catalog Number:10-2626Activity:c-MET and ALK inhibitorChemical Name:3-[(1R)-1-(2,6-Dichloro-3-fluorophenyl)ethoxy]-5-[1-(4-piperidinyl)-1H-pyrazol-4-yl]-2-pyridinamineAlternate Names:PF-02341066, PF-1066Molecular Weight:450.34Molecular Formula:C21H22Cl2FN5OSolubility:Soluble in DMSO (up to 25 mg/ml with warming) or in Ethanol (up to 25 mg/ml with warming)Physical Properties:White solidPurity:98% by HPLC
NMR (Conforms)Storage Temperature:-20°CStability:Stable for 1 year from date of purchase as supplied. Solutions in DMSO or ethanol may be stored at -20°C for up to 2 months.Shipping Code:RT -
CUDC-101 | Dual HDAC and EGFR inhibitor
From $70.00CAS:1012054-59-9Catalog Number:10-2491Activity:Dual HDAC and EGFR inhibitorChemical Name:7-((4-((3-Ethynylphenyl)amino)-7-methoxyquinazolin-6-yl)oxy)-N-hydroxyheptanamideMolecular Weight:434.49Molecular Formula:C24H26N4O4Solubility:Soluble in DMSO (up to 25 mg/ml)Physical Properties:White or off-white solidPurity:99% by HPLC
NMR (Conforms)Storage Temperature:-20°CStability:Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 1 month.Shipping Code:RT -
CZC-8004 | Pan-kinase inhibitor
From $90.00CAS:916603-07-1Catalog Number:10-3032Activity:Multi-kinase inhibitor; affinity ligandChemical Name:N2-[4-(Aminomethyl)phenyl]-5-fluoro-N4-phenyl-2,4-[yrimidinediamineMolecular Weight:309.33Molecular Formula:C17H16FN5Solubility:Soluble in DMSO (up to 30 mg/ml) or in Ethanol (up to 2.5 mg/ml with warming)Physical Properties:Off-white solidPurity:98% by TLC
NMR (Conforms)Storage Temperature:-20°Stability:Stable for 1 year from date of purchase as supplied. Solutions in DMSO or ethanol may be stored at -20° for up to 3 months.Shipping Code:RT
EXPLORE OTHER Cancer
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