Highly Selective Inhibitors
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GSK2656157 | PERK inhibitor
From $40.00CAS:1337532-29-2Catalog Number:10-4855Activity:PERK inhibitorChemical Names:1-[5-(4-Amino-7-methylpyrrolo[2,3-d]pyrimidin-5-yl)-4-fluoro-2,3-dihydroindol-1-yl]-2-(6-methylpyridin-2-yl)ethanoneMolecular Weight:416.45Molecular Formula:C23H21FN6OSolubility:Soluble in DMSO (10 mg/ml with warming)Physical Properties:White solidPurity:>98% HPLC
NMR (Conforms)Storage Temperature:-20°CStability:Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 1 month.Shipping Code:RT -
GSK583 | RIP2 kinase inhibitor
From $40.00CAS:1346547-00-9Catalog Number:10-4761Activity:RIP2 kinase inhibitorChemical Name:6-tert-Butylsulfonyl-N-(5-fluoro-1H-indazol-3-yl)quinoline-4-amineMolecular Weight:398.45Molecular Formula:C20H19FN4O2SSolubility:Soluble in DMSO (up to at least 25 mg/ml).Physical Properties:Pale yellow solidPurity:98% by HPLC
NMR (Conforms)Storage Temperature:-20°Stability:Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20° for up to 1 month.Shipping Code:RT -
Idelalisib | Selective PI3Kδ Inhibitor
From $60.00CAS:870281-82-6Catalog Number:10-4820Activity:Selective PI3Kδ InhibitorChemical Name:5-Fluoro-3-phenyl-2-[(1S)-1-(7H-purin-6-ylamino)propyl]quinazolin-4-oneAlternate Names:CAL-101Molecular Weight:415.43Molecular Formula:C21H18FN7OSolubility:Soluble in DMSO (>25 mg/ml)Physical Properties:White solidPurity:>98% by HPLC
NMR (Conforms)Storage Temperature:-20°CStability:Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 2 months.Shipping Code:RT -
Imatinib mesylate | BCR-ABL inhibitor
From $30.00CAS:220127-57-1Catalog Number:10-1060Activity:BCR-ABL inhibitorAlternate Names:GleevecChemical Name:4-[(4-Methyl-1-piperazinyl)methyl]-N-[4-methyl-3-[[4-(3-pyridinyl)-2-pyrimidinyl]amino]phenyl]benzamide methanesulfonateMolecular Weight:589.73Molecular Formula:C29H31N7O CH3SO3HSolubility:Soluble in DMSO (up to 50 mg/ml) or in Water (up to 50 mg/ml).Physical Properties:White solidPurity:98% by TLC
NMR (Conforms)Storage Temperature:-20°CStability:Stable for 1 year from date of purchase as supplied. Solutions in DMSO or water may be stored at -20°C for up to 3 months.Shipping Code:RT -
Intelliscreen™ Highly-Selective Kinase Inhibitor Library
$3,700.00Catalog Number:10-7001Description:166 highly selective inhibitors of various kinases.Solubility:DMSOSupplied As:DSMO solution @ 10mMStorage Temperature:-80°CStability:Stable for up to 1 year when stored as supplied @ -80°CPrice:$3 700.00
