Highly Selective Inhibitors
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NU7441 | DNA-PK inhibitor
From $40.00CAS:503468-95-9Catalog Number:10-4810Activity:DNA-PK inhibitorChemical Name:8-Dibenzothiophen-4-yl-2-morpholin-4-ylchromen-4-oneAlternate Name:Ku-57788Molecular Weight:413.49Molecular Formula:C25H19NO3SSolubility:Soluble in DMSO (up to 10 mg/ml with warming).Physical Properties:Off-white to beige solidPurity:98% by TLC
NMR (Conforms)Storage Temperature:-20°Stability:Stable for 1 year as supplied. Solutions in DMSO may be stored at -20° for up to 3 months.Shipping Code:RT -
NVP-BGJ398 | Pan-specific FGFR inhibitor
From $65.00CAS:872511-34-7Catalog Number:10-4817Activity:Pan-specific FGFR inhibitorChemical Name:3-(2,6-Dichloro-3,5-dimethoxyphenyl)-1-(6-{[4-(4-ethyl-1-piperazinyl)phenyl]amino}-4-pyrimidinyl)-1-methylureaAlternate Names:InfigratinibMolecular Weight:560.48Molecular Formula:C26H31Cl2N7O3Solubility:Soluble in DMSO (up to 5 mg/ml)Physical Properties:White solidPurity:98% by HPLC
NMR (Conforms)Storage Temperature:-20°CStability:Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 2 months.Shipping Code:RT -
PLX5622 | Highly selective CSF1R inhibitor
From $70.00CAS:1303420-67-8Catalog Number:10-4726Activity:Highly selective CSF1R inhibitorChemical Names:6-Fluoro-N-[(5-fluoro-2-methoxypyridin-3-yl)methyl]-5-[(5-methyl-1H-pyrrolo[2,3-b]pyridine-3-yl)methyl]pyridine-2-amineMolecular Weight:395.41Molecular Formula:C21H19F2N5OSolubility:Soluble in DMSO (>25 mg/ml)Physical Properties:Pale yellow solidPurity:>98% HPLC
NMR (Conforms)Storage Temperature:-20°CStability:Stable for 2 years from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 3 months.Shipping Code:RT -
Quizartinib | Selective FLT3 Inhibitor
From $50.00CAS:950769-58-1Catalog Number:10-4813Activity:Selective FLT3 inhibitorChemical Name:1-(5-(t-Butyl)isoxazol-3-yl)-3-(4-(7-(2-morpholinoethoxy)benzo[d]imidazo[2,1-b]thiazol-2-yl)phenyl)ureaAlternate Names:AC220Molecular Weight:560.67Molecular Formula:C29H32N6O4SSolubility:Soluble in DMSO (up to at least 25 mg/ml)Physical Properties:Off-white solidPurity:98% by HPLC
NMR (Conforms)Storage Temperature:-20°CStability:Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 1 month.Shipping Code:RT
