Kinases Archives

R428 | Potent and selective AXL inhibitor

CAS:

1037624-75-1

Catalog Number:

10-4676

Activity:

Potent and selective AXL inhibitor

Chemical Name:

1-(3,4-Diazatricyclo[9.4.0.02,7]pentadeca-1(15),2,4,6,11,13-hexaen-5-yl)-3-N-[(7S)-7-pyrrolidin-1-yl-6,7,8,9-tetrahydro-5H-benzo[7]annulen-3-yl]-1,2,4-triazole-3,5-diamine

Alternate Names:

Bemcentinib; BGB324

Molecular Weight:

506.64

Molecular Formula:

C₃₀H₃₄N₈

Solubility:

Soluble in DMSO (up to at least 25 mg/ml)

Physical Properties:

Yellow solid

Purity:

98% by HPLC
NMR (Conforms)

Storage Temperature:

-20°C

Stability:

Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 3 months.

Shipping Code:

RT

From $75.00
View Product This product has multiple variants. The options may be chosen on the product page
Rebastinib | Bcl-Abl1 inhibitor

CAS:
1020172-07-9
Catalog Number:
10-4689
View Product This product has multiple variants. The options may be chosen on the product page
Ribociclib | CDK4/6 inhibitor

CAS:

1211441-98-3

Catalog Number:

10-4807

Activity:

CDK4/6 inhibitor

Chemical Name:

7-Cyclopentyl-N,N-dimethyl-2-((5-(piperazin-1-yl)pyridin-2-yl)amino)-7H-pyrrolo[2,3-d]pyrimidine-6-carboxamide

Alternate Names:

LEE011

Molecular Weight:

434.54

Molecular Formula:

C₂₃H₃₀N₈O₃

Solubility:

Soluble in DMSO (up to 10 mg/ml)

Physical Properties:

Off-white solid

Purity:

98% by HPLC
NMR (Conforms)

Storage Temperature:

-20°C

Stability:

Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 2 months.

Shipping Code:

RT

From $60.00
View Product This product has multiple variants. The options may be chosen on the product page
RO-3306 | Selective CDK1 inhibitor

CAS:

872573-93-8

Catalog Number:

10-4126

Activity:

Selective CDK1 inhibitor

Chemical Name:

5-(6-Quinolinylmethylene)-2-[(2-thienylmethyl)amino]-4(5H)-thiazolone

Molecular Weight:

351.45

Molecular Formula:

C₁₈H₁₃N₃OS₂

Solubility:

Soluble in DMSO (up to 15 mg/ml)

Physical Properties:

Off-white or pale yellow solid

Purity:

98% by HPLC
NMR (Conforms)

Storage Temperature:

-20°C

Stability:

Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 3 months.

Shipping Code:

RT

From $65.00
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Roscovitine | p34/cdc2 inhibitor

CAS:

186692-46-6

Catalog Number:

10-1332

Activity:

p34/cdc2 inhibitor

Chemical Name:

(R)-2-((6-(Benzylamino)-9-isopropyl-9H-purin-2-yl)amino)butan-1-ol

Molecular Weight:

354.46

Molecular Formula:

C₁₉H₂₆N₆O

Solubility:

Soluble in DMSO (up to 10 mg/ml, with warming) or in Ethanol (up to 10 mg/ml).

Physical Properties:

White solid

Purity:

99% by TLC
NMR (Conforms)

Storage Temperature:

-20°C

Stability:

Stable for 2 years from date of purchase as supplied. Solutions in DMSO or ethanol may be stored at -20° for up to 3 months.

Shipping Code:

RT

From $45.00
View Product This product has multiple variants. The options may be chosen on the product page

Kinases

R428 | Potent and selective AXL inhibitor

Rebastinib | Bcl-Abl1 inhibitor

Ribociclib | CDK4/6 inhibitor

RO-3306 | Selective CDK1 inhibitor

Roscovitine | p34/cdc2 inhibitor

EXPLORE OTHER Cancer

20% OFF

Focus Biomolecules • Plymouth Meeting, PA USA • 1-855-FOCUS21

Focus Biomolecules
Plymouth Meeting, PA USA
1-855-FOCUS21

Kinases

R428 | Potent and selective AXL inhibitor

Rebastinib | Bcl-Abl1 inhibitor

Ribociclib | CDK4/6 inhibitor

RO-3306 | Selective CDK1 inhibitor

Roscovitine | p34/cdc2 inhibitor

EXPLORE OTHER Cancer

20% OFF

Focus Biomolecules • Plymouth Meeting, PA USA • 1-855-FOCUS21

Focus Biomolecules Plymouth Meeting, PA USA1-855-FOCUS21

Focus Biomolecules
Plymouth Meeting, PA USA
1-855-FOCUS21