Kinases
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Ruxolitinib | JAK inhibitor
From $65.00CAS:941678-49-5Catalog Number:10-4511Activity:JAK inhibitorAlternate Names:INCB 018424Chemical Name:βR-Cyclopentyl-4-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-1H-pyrazole-1-propanenitrileMolecular Weight:306.37Molecular Formula:C17H18N6Solubility:Soluble in DMSO (up to 28 mg/ml) or in Ethanol (up to 15 mg/ml with warming).Physical Properties:White solidPurity:99% by HPLC
NMR (Conforms)Storage Temperature:-20°Stability:Stable for 1 year from date of purchase as supplied. Solutions in DMSO or ethanol may be stored at -20° for up to 3 months.Shipping Code:RT -
Saracatinib | Src family kinase inhibitor
From $40.00CAS:379231-04-6Catalog Number:10-2901Activity:Src family kinase inhibitorChemical Names:N-(5-Chloro-1,3-benzodioxol-4-yl)-7-[2-(4-methyl-1-piperazinyl)ethoxy]-5-[(tetrahydro-2H-pyran-4-yl)oxy]-4-quinazolinamine; AZD0530Molecular Weight:542.03Molecular Formula:C27H32ClN5O5Solubility:Soluble in DMSO (50 mg/ml) and ethanol (54 mg/mL with warming)Physical Properties:White solidPurity:>98% HPLC
NMR (Conforms)Storage Temperature:-20°CStability:Stable for 2 years from date of purchase as supplied. Solutions in DMSO or ethanol may be stored at -20°C for up to 3 months.Shipping Code:RT -
SB-525334 | ALK5 inhibitor
From $60.00CAS:356559-20-1Catalog Number:10-2983Activity:ALK5 (TGFβR1) inhibitorChemical Name:6-[2-(1,1-Dimethylethyl)-5-(6-methyl-2-pyridinyl)-1H-imidazol-4-yl]quinoxalineMolecular Weight:343.42Molecular Formula:C21H21N5Solubility:Soluble in DMSO (up tp 30 mg/ml)Physical Properties:Yellow solidPurity:98% by HPLC
NMR (Conforms)Storage Temperature:-20°CStability:Stable for 2 years from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 3 months.Shipping Code:RT -
SBI-0206965 | ULK1 inhibitor
From $65.00CAS:1884220-36-3Catalog Number:10-1623Activity:ULK1 inhibitorChemical Name:2-((5-Bromo-2-((3,4,5-trimethoxyphenyl)amino)pyrimidin-4-yl)oxy)-N-methylbenzamideMolecular Weight:489.32Molecular Formula:C21H21BrN4O4Solubility:Soluble in DMSO (up to 30 mg/ml)Physical Properties:White solidPurity:98% by HPLC/TLC
NMR (Conforms)Storage Temperature:-20°CStability:Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 3 months.Shipping Code:RT -
Selonsertib | ASK1 inhibitor
From $50.00CAS:1448428-04-3Catalog Number:10-4696Activity:ASK1 inhibitorChemical Names:5-(4-Cyclopropylimidazol-1-yl)-2-fluoro-4-methyl-N-[6-(4-propan-2-yl)-1,2,4-triazol-3-yl)pyridine-2-yl]benzamideAlternate Name:GS-4997Molecular Weight:445.50Molecular Formula:C24H24FN7OSolubility:Soluble in DMSO (>25 mg/ml)Physical Properties:White solidPurity:>98% HPLC
NMR (Conforms)Storage Temperature:-20°CStability:Stable for 2 years from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 3 months.Shipping Code:RT
EXPLORE OTHER Cancer
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- p53 & Other Tumor Suppressors
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