Kinases
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Sorafenib | Multi-kinase inhibitor
From $40.00CAS:284461-73-0Catalog Number:10-2174Activity:Inhibitor of Raf-1 and other kinasesAlternate Names:BAY 43-9006Chemical Name:4-(4-(3-(4-chloro-3-(trifluoromethyl)phenyl)ureido)phenoxy)-N-methylpicolinamideMolecular Weight:464.83Molecular Formula:C21H16ClF3N4O3Solubility:Soluble in DMSO (up to 200 mg/ml) or in Ethanol (up to 3 mg/ml).Physical Properties:Off-white solidPurity:99% by TLC
NMR (Conforms)Storage Temperature:-20°Stability:Stable for 2 years from date of purchase as supplied. Solutions in DMSO or ethanol may be stored at -20° for up to 1 month.Shipping Code:RT -
SU-1498 | VEGFR kinase inhibitor
From $55.00CAS:168835-82-3Catalog Number:10-2074Activity:VEGFR kinase inhibitorChemical Name:(E)-N-(3′-Phenylpropyl)-α-cyano-3′,5′-diisopropyl-4′-hydroxycinnamamideMolecular Weight:390.52Molecular Formula:C25H30N2O2Solubility:Soluble in DMSO.Physical Properties:Pale yellow solidPurity:>98% TLC
NMR (Conforms)Storage Temperature:-20°Stability:Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20° for up to 3 months.Shipping Code:RT -
SU-5402 | FGFR Phosphorylation inhibitor
From $70.00CAS:215543-92-3Catalog Number:10-2520Activity:FGFR Phosphorylation inhibitorAlternate Names:PF-02969207Chemical Name:3-[4-Methyl-2-(2-oxo-1,2-dihydro-indol-3-ylidenemethyl)-1H-pyrrol-3-yl]-propionic acidMolecular Weight:296.32Molecular Formula:C17H16N2O3Solubility:Soluble in DMSO (up to 10 mg/ml).Physical Properties:Orange solidPurity:98% by HPLC
NMR (Conforms)Storage Temperature:-20°Stability:Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20° for up to 3 months.Shipping Code:RT -
SU9516 | pan-specific CDK inhibitor
From $75.00CAS:SU9516Catalog Number:10-5705Activity:pan-specific CDK inhibitorChemical Names:(Z)-1,3-Dihydro-3-(1H-imidazol-4-ylmethylene)-5-methoxy-2H-2-oneMolecular Weight:241.25Molecular Formula:C13H11N3O2Solubility:Soluble in DMSO (25 mg/ml)Physical Properties:Orange solidPurity:>98% HPLC
NMR (Conforms)Storage Temperature:-20°CStability:Stable for 2 years from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 2 months.Shipping Code:RT -
Sunitinib malate | VEGFR, PDGFR kinase inhibitor
From $60.00CAS:341031-54-7Catalog Number:10-1078Activity:VEGFR, PDGFR kinase inhibitorAlternate Names:SU-11248Chemical Name:N-[2-(Diethylamino)ethyl]-5-[(Z)-(5-fluoro-1,2-dihydro-2-oxo-3H-indol-3-ylidene)methyl]-2,4-dimethyl-1H-pyrrole-3-carboxamide malateMolecular Weight:532.57Molecular Formula:C22H27FN4O4 C4H6O5Solubility:Soluble in DMSO (up to 13 mg/ml).Physical Properties:Orange solidPurity:98% by TLC
NMR (Conforms)Storage Temperature:-20°CStability:Stable for 2 years from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 3 months.Shipping Code:RT
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