Kinases
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DRB | Transcription inhibitor/CK2 inhibitor
From $27.00CAS:53-85-0Catalog Number:10-2047Activity:Transcription inhibitor, CK2 inhibitorChemical Name:5,6-Dichloro-1-β-D-ribofuranosylbenzimidazoleAlternate Names:5,6-Dichlorobenzimidazole riboside; NSC 401575Molecular Weight:319.14Molecular Formula:C12H12Cl2N2O4Solubility:Soluble in DMSO (up to 20 mg/ml)Physical Properties:White solidPurity:98% by HPLC
NMR (Conforms)Storage Temperature:-20°CStability:Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 3 months.Shipping Code:RT -
Duvelisib | PI3Kdelta/gamma inhibitor
From $65.00CAS:1201438-56-3Catalog Number:10-4788Activity:PI3Kδ/γ inhibitor/Cancer immunotherapy enhancerChemical Name:8-Chloro-2-phenyl-3-[(1S)-1-(7H-purin-6-ylamino)ethyl]isoquinolin-1-oneAlternative Name:IPI-145Molecular Weight:416.87Molecular Formula:C22H17ClN6OSolubility:Soluble in DMSO (up to at least 25 mg/ml)Physical Properties:White solidPurity:98% by HPLC
NMR (Conforms)Storage Temperature:-20°CStability:Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 3 months.Shipping Code:RT -
ERGi-USU | Highly Selective ERG Inhibitor
From $35.00CAS:1147-56-4Catalog Number:10-4290Activity:Highly selective ERG inhibitorChemical Name:1-(2-Thiazolylazo)-2-naphtholAlternate Names:NSC139021Molecular Weight:255.30Molecular Formula:C13H9N3OSSolubility:Soluble in DMSO (up to at least 10 mg/ml)Physical Properties:Red or orange solidPurity:98% by TLC
NMR (Conforms)Storage Temperature:-20°CStability:Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 1 month.Shipping Code:RT
EXPLORE OTHER Cancer
- ADC warheads
- Angiogenesis
- Autophagy
- Cancer Cell Metabolism
- Cancer Stem Cells
- Cell Cycle
- Cellular Stress
- Chemotherapeutics
- Cytoskeleton
- DNA Damage/Repair
- Drug resistance
- Epigenetics
- Gene Regulation/Transcription
- Growth factors
- Immuno-oncology
- Metastasis
- Other Cancer
- p53 & Other Tumor Suppressors
- Programmed cell death
- Stem Cells
- Ubiquitin proteasome
- Wnt/ß-Catenin
