Kinases Archives

Purvalanol A | CDK inhibitor

CAS:

212844-53-6

Catalog Number:

10-2868

Activity:

CDK Inhibitor

Chemical Name:

(2R)-2-[[6-[(3-Chlorophenyl)amino]-9-(1-methylethyl)-9H-purin-2-yl]amino]-3-methyl-1-butanol

Alternate Names:

NG-60

Molecular Weight:

388.89

Molecular Formula:

C₁₉H₂₅ClN₆O

Solubility:

Soluble in DMSO (up to 35 mg/ml)

Physical Properties:

Pale green solid

Purity:

98% by HPLC
NMR (Conforms)

Storage Temperature:

-20°C

Stability:

Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 2 months.

Shipping Code:

RT

From $50.00
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PX-866 | PI3-K inhibitor

CAS:

502632-66-8

Catalog Number:

10-1315

Activity:

PI3-K inhibitor

Molecular Weight:

525.6

Molecular Formula:

C₂₉H₃₅NO₈

Solubility:

Soluble in DMSO (up to 25 mg/ml).

Physical Properties:

Orange solid

Purity:

98% by TLC
NMR (Conforms)

Storage Temperature:

-20°C

Stability:

Stable for 2 years from date of purchase as supplied. Solutions in DMSO may be stored at -20° for up to 2 months.

Shipping Code:

RT

From $60.00
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Quizartinib | Selective FLT3 Inhibitor

CAS:

950769-58-1

Catalog Number:

10-4813

Activity:

Selective FLT3 inhibitor

Chemical Name:

1-(5-(t-Butyl)isoxazol-3-yl)-3-(4-(7-(2-morpholinoethoxy)benzo[d]imidazo[2,1-b]thiazol-2-yl)phenyl)urea

Alternate Names:

AC220

Molecular Weight:

560.67

Molecular Formula:

C₂₉H₃₂N₆O₄S

Solubility:

Soluble in DMSO (up to at least 25 mg/ml)

Physical Properties:

Off-white solid

Purity:

98% by HPLC
NMR (Conforms)

Storage Temperature:

-20°C

Stability:

Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 1 month.

Shipping Code:

RT

From $50.00
View Product This product has multiple variants. The options may be chosen on the product page
R428 | Potent and selective AXL inhibitor

CAS:

1037624-75-1

Catalog Number:

10-4676

Activity:

Potent and selective AXL inhibitor

Chemical Name:

1-(3,4-Diazatricyclo[9.4.0.02,7]pentadeca-1(15),2,4,6,11,13-hexaen-5-yl)-3-N-[(7S)-7-pyrrolidin-1-yl-6,7,8,9-tetrahydro-5H-benzo[7]annulen-3-yl]-1,2,4-triazole-3,5-diamine

Alternate Names:

Bemcentinib; BGB324

Molecular Weight:

506.64

Molecular Formula:

C₃₀H₃₄N₈

Solubility:

Soluble in DMSO (up to at least 25 mg/ml)

Physical Properties:

Yellow solid

Purity:

98% by HPLC
NMR (Conforms)

Storage Temperature:

-20°C

Stability:

Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 3 months.

Shipping Code:

RT

From $75.00
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Ribociclib | CDK4/6 inhibitor

CAS:

1211441-98-3

Catalog Number:

10-4807

Activity:

CDK4/6 inhibitor

Chemical Name:

7-Cyclopentyl-N,N-dimethyl-2-((5-(piperazin-1-yl)pyridin-2-yl)amino)-7H-pyrrolo[2,3-d]pyrimidine-6-carboxamide

Alternate Names:

LEE011

Molecular Weight:

434.54

Molecular Formula:

C₂₃H₃₀N₈O₃

Solubility:

Soluble in DMSO (up to 10 mg/ml)

Physical Properties:

Off-white solid

Purity:

98% by HPLC
NMR (Conforms)

Storage Temperature:

-20°C

Stability:

Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 2 months.

Shipping Code:

RT

From $60.00
View Product This product has multiple variants. The options may be chosen on the product page

Kinases

Purvalanol A | CDK inhibitor

PX-866 | PI3-K inhibitor

Quizartinib | Selective FLT3 Inhibitor

R428 | Potent and selective AXL inhibitor

Ribociclib | CDK4/6 inhibitor

EXPLORE OTHER Cancer

Focus Biomolecules • Plymouth Meeting, PA USA • 1-855-FOCUS21

Focus Biomolecules
Plymouth Meeting, PA USA
1-855-FOCUS21

Kinases

Purvalanol A | CDK inhibitor

PX-866 | PI3-K inhibitor

Quizartinib | Selective FLT3 Inhibitor

R428 | Potent and selective AXL inhibitor

Ribociclib | CDK4/6 inhibitor

EXPLORE OTHER Cancer

Focus Biomolecules • Plymouth Meeting, PA USA • 1-855-FOCUS21

Focus Biomolecules Plymouth Meeting, PA USA1-855-FOCUS21

Focus Biomolecules
Plymouth Meeting, PA USA
1-855-FOCUS21