BiochemicalTargets

Approved Drugs

Drugs approved by the FDA or other agencies for use in medicine are excellent tools for research because they are demonstrated to have good absorption (bioavailable), distribution and activity, and pharmacokinetics for use in vivo experiments. They are used in cells or animals for basic research, and for drug discovery (repurposing, benchmarking and other applications).

  • Carfilzomib | Proteasome inhibitor

    CAS:
    868540-17-4
    Catalog Number:
    10-1477
    Activity:
    Proteasome inhibitor
    Alternate Names:
    PR-171
    Chemical Name:
    (αS)-α-[[2-(4-morpholinyl)acetyl]amino]benzenebutanoyl-L-leucyl-N-[(1S)-3-methyl-1-[[(2R)-2-methyl-2-oxiranyl]carbonyl]butyl]- L-Phenylalaninamide
    Molecular Weight:
    719.93
    Molecular Formula:
    C40H57N5O7
    Solubility:
    Soluble in DMSO (up to 80 mg/ml) or in Ethanol (up to 25 mg/ml).
    Physical Properties:
    White solid
    Purity:
    98% by TLC
    NMR (Conforms)
    Storage Temperature:
    -20°
    Stability:
    Stable for 1 year from date of purchase as supplied. Solutions in DMSO or ethanol may be stored at -20° for up to 1 week.
    Shipping Code:
    RT
    From $50.00
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  • Chloroquine phosphate | Antimalarial/Autophagy inhibitor

    CAS:
    50-63-5
    Catalog Number:
    10-2473
    Activity:
    Antimalarial/Autophagy inhibitor
    Chemical Names:
    N4-(7-Chloro-4-quinolinyl)-N1,N1-dimethyl-1,4-pentanediamine, diphosphate
    Molecular Weight:
    515.87
    Molecular Formula:
    C18H26ClN3·2H3PO4
    Solubility:
    Soluble in Water (25 mg/ml)
    Physical Properties:
    White solid
    Purity:
    98% TLC
    NMR (Conforms)
    Storage Temperature:
    -20°C
    Stability:
    Stable for 2 years from date of purchase as supplied. Solutions in water may be stored at -20°C for up to 3 months.
    Shipping Code:
    RT
    From $25.00
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  • Cilostazol | PDE3A inhibitor

    CAS:
    73963-72-1
    Catalog Number:
    10-1131
    Activity:
    PDE3A inhibitor
    Chemical Name:
    6-[4-(1-Cyclohexyl-1H-tetrazol-5-yl)-butoxy]-3,4-dihydro-2(1H)-quinolinone
    Molecular Weight:
    369.46
    Molecular Formula:
    C20H27N5O2
    Solubility:
    Soluble in DMSO (up to 20 mg/ml).
    Physical Properties:
    White solid
    Purity:
    98% by TLC
    NMR (Conforms)
    Storage Temperature:
    RT
    Stability:
    Stable for 2 years from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 2 months
    Shipping Code:
    RT
    From $40.00
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  • Cinacalcet | Calcium sensing receptor (CaSR) agonist

    CAS:
    364782-34-3
    Catalog Number:
    10-2957
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  • Cisplatin | Anticancer agent

    CAS:
    15663-27-1
    Catalog Number:
    10-2204
    Activity:
    Anticancer agent
    Chemical Name:
    Cis-Diaminodichloroplatinum
    Alternate Names:
    CDDP; cis-Diamineplatinum(II) dichloride
    Molecular Weight:
    300.05
    Molecular Formula:
    Cl2H4N2Pt
    Solubility:
    Soluble in Water (up to 2.5 mg/ml with warming)
    Physical Properties:
    Yellow solid
    Purity:
    98% by HPLC
    Elemental Analysis (Conforms)
    Storage Temperature:
    RT
    Stability:
    Stable for 1 year from date of purchase as supplied. Solutions in distilled water are not stable and must be used within 1 working day. do not store solutions.
    Shipping Code:
    RT
    From $50.00
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  • Citalopram HBr | Serotonin uptake inhibitor

    CAS:
    59729-32-7
    Catalog Number:
    10-2458
    Activity:
    Serotonin uptake inhibitor
    Chemical Name:
    1-[3-(Dimethylamino)propyl]-1-(4-fluorophenyl)-1,3-dihydro-5-isobenzofurancarbonitrile hydrobromide
    Molecular Weight:
    405.31
    Molecular Formula:
    C20H21FN2O HBr
    Solubility:
    Soluble in Water (up to 4 mg/ml), DMSO (up to 25 mg/ml) or in Ethanol (up to 20 mg/ml)
    Physical Properties:
    White solid
    Purity:
    98% by TLC
    NMR (Conforms)
    Storage Temperature:
    -20°C
    Stability:
    Stable for 2 years from date of purchase as supplied. Solutions in water, DMSO or ethanol may be stored at -20°C for up to 2 months.
    Shipping Code:
    RT
    From $52.00
    View Product This product has multiple variants. The options may be chosen on the product page
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