Approved Drugs
Drugs approved by the FDA or other agencies for use in medicine are excellent tools for research because they are demonstrated to have good absorption (bioavailable), distribution and activity, and pharmacokinetics for use in vivo experiments. They are used in cells or animals for basic research, and for drug discovery (repurposing, benchmarking and other applications).
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Captopril | Angiotensin-converting enzyme inhibitor
From $30.00CAS:62571-86-2Catalog Number:10-2253Activity:Angiotensin-converting enzyme inhibitorChemical Name:(2S)-1-(3-Mercapto-2-methyl-propionyl)-L-prolineMolecular Weight:217.28Molecular Formula:C9H15NO3SSolubility:Soluble in DMSO (up to 20 mg/ml) or in Water (up to 20 mg/ml).Physical Properties:White solidPurity:98% by HPLC
NMR (Conforms)Storage Temperature:-20°CStability:Stable for 1 year from date of purchase as supplied. Solutions in DMSO or distilled water may be stored at -20°C for up to 1 monthShipping Code:RT -
Carfilzomib | Proteasome inhibitor
From $50.00CAS:868540-17-4Catalog Number:10-1477Activity:Proteasome inhibitorAlternate Names:PR-171Chemical Name:(αS)-α-[[2-(4-morpholinyl)acetyl]amino]benzenebutanoyl-L-leucyl-N-[(1S)-3-methyl-1-[[(2R)-2-methyl-2-oxiranyl]carbonyl]butyl]- L-PhenylalaninamideMolecular Weight:719.93Molecular Formula:C40H57N5O7Solubility:Soluble in DMSO (up to 80 mg/ml) or in Ethanol (up to 25 mg/ml).Physical Properties:White solidPurity:98% by TLC
NMR (Conforms)Storage Temperature:-20°Stability:Stable for 1 year from date of purchase as supplied. Solutions in DMSO or ethanol may be stored at -20° for up to 1 week.Shipping Code:RT -
Chloroquine phosphate | Antimalarial/Autophagy inhibitor
From $25.00CAS:50-63-5Catalog Number:10-2473Activity:Antimalarial/Autophagy inhibitorChemical Names:N4-(7-Chloro-4-quinolinyl)-N1,N1-dimethyl-1,4-pentanediamine, diphosphateMolecular Weight:515.87Molecular Formula:C18H26ClN3·2H3PO4Solubility:Soluble in Water (25 mg/ml)Physical Properties:White solidPurity:98% TLC
NMR (Conforms)Storage Temperature:-20°CStability:Stable for 2 years from date of purchase as supplied. Solutions in water may be stored at -20°C for up to 3 months.Shipping Code:RT -
Chloroquine phosphate | autophagy inhibitor
From $25.00CAS:50-63-5Catalog Number:10-2473Activity:autophagy inhibitorChemical Name:N4-(7-Chloro-4-quinolinyl)-N1,N1-dimethyl-1,4-pentanediamine, diphosphateMolecular Weight:515.87Molecular Formula:C18H26ClN3·2H3PO4Solubility:Soluble in Water (up to 25 mg/ml).Physical Properties:White solidPurity:98% by TLC
NMR (Conforms)Storage Temperature:RTStability:Stable for 2 years from date of purchase as supplied. Solutions in distilled water may be stored at -20° for up to 3 months.Shipping Code:RT -
Cilostazol | PDE3A inhibitor
From $40.00CAS:73963-72-1Catalog Number:10-1131Activity:PDE3A inhibitorChemical Name:6-[4-(1-Cyclohexyl-1H-tetrazol-5-yl)-butoxy]-3,4-dihydro-2(1H)-quinolinoneMolecular Weight:369.46Molecular Formula:C20H27N5O2Solubility:Soluble in DMSO (up to 20 mg/ml).Physical Properties:White solidPurity:98% by TLC
NMR (Conforms)Storage Temperature:RTStability:Stable for 2 years from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 2 monthsShipping Code:RT
