Intelliscreen™ Protease Inhibitors Mini-Library

The IntelliscreenTM Protease Inhibitor mini-library is a useful screening tool for determining protease family involvement during proteolysis. The inhibitors have been selected to cover the most common protease families involved in degradation and / or processing, including aspartic, cysteine, serine, etc. peptidases; caspases; proteasome; metalloproteases; aminopeptidases, secretases, and signal peptide peptidases; and more.

Catalog Number:
10-7340
Description:
25 protease inhibitors covering the most common families
Solubility:
DMSO
Supplied As:
DMSO solution @ 10mM
Storage Temperature:
-80°C
Stability:
Stable for up to 1 year when stored as supplied @ -80°C
Price:
$600.00
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Please note that we do not sell to individuals and that all orders placed by non-research organizations will incur a $20 restocking/refund fee

View Product Datasheet
MSDS

  • 1,10-Phenanthroline HCl | Zn metalloprotease inhibitor

    CAS:
    18851-33-7
    Catalog Number:
    10-3017
    Activity:
    Zn metalloprotease inhibitor
    Alternate Names:
    o-Phenanthroline hydrochloride hydrate
    Molecular Weight:
    234.68
    Molecular Formula:
    C13H8N2 • HCl &bul; H2O
    Solubility:
    Soluble in DMSO (up to 5 mg/ml) or in Water (up to 2 mg/ml)
    Physical Properties:
    White solid
    Purity:
    98% by TLC
    NMR (Conforms)
    Storage Temperature:
    RT
    Stability:
    Stable for 2 year from date of purchase as supplied. Solutions in DMSO or distilled water may be stored at -20°C for up to 3 months.
    Shipping Code:
    RT
    From $20.00
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  • 1G244 | DPP8/9 inhibitor

    CAS:
    847928-32-9
    Catalog Number:
    10-4584
    Activity:
    DPP8/9 inhibitor
    Chemical Names:
    (S)-2-Amino-4-{4-[bis-(4-fluorophenyl)-methyl]piperazin-1-yl}-1-(1,3-dihydro-isoindol-2-yl)-butane-1,4-dione
    Alternate Name:
    PTX-1210
    Molecular Weight:
    504.57
    Molecular Formula:
    C29H30F2N4O2
    Solubility:
    Soluble in DMSO (>20 mg/ml)
    Physical Properties:
    Off-white solid
    Purity:
    >98% HPLC
    NMR (Conforms)
    Storage Temperature:
    -20°C
    Stability:
    Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 2 months.
    Shipping Code:
    RT
    From $70.00
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  • AEBSF HCl | Protease inhibitor

    CAS:
    30827-99-7
    Catalog Number:
    10-1348
    Activity:
    Protease inhibitor
    Chemical Name:
    4-(2-Aminoethyl)benzenesulfonyl fluoride hydrochloride
    Molecular Weight:
    239.69
    Molecular Formula:
    C8H10FNO2S • HCl
    Solubility:
    Soluble in DMSO (up to 25 mg/ml) or in Water (up to 100 mg/ml)
    Physical Properties:
    White solid
    Purity:
    98%
    NMR (Conforms)
    Storage Temperature:
    -20°C
    Stability:
    Stable for 1 year from date of purchase as supplied. Solutions at pH <7 are stable for up to 6 months if stored in the refrigerator
    Shipping Code:
    RT
    From $42.00
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  • ALLM | Calpain inhibitor

    CAS:
    136632-32-1
    Catalog Number:
    10-1349
    Activity:
    Calpain inhibitor
    Chemical Name:
    N-Acetyl-Leu-Leu-Methional
    Alternate Names:
    Ac-LLM-CHO
    Molecular Weight:
    401.56
    Molecular Formula:
    C19H35N3O4S
    Solubility:
    Soluble in DMSO (up to 10 mg/ml) or in Ethanol (up to 5 mg/ml).
    Physical Properties:
    White solid
    Purity:
    98% by HPLC
    NMR (Conforms)
    Storage Temperature:
    -20°C
    Stability:
    Stable for 1 year from date of purchase as supplied. Solutions in DMSO or ethanol may be stored at -20°C for up to 1 month.
    Shipping Code:
    RT
    From $60.00
    View Product This product has multiple variants. The options may be chosen on the product page

  • ALLN | Calpain inhibitor

    CAS:
    110044-82-1
    Catalog Number:
    10-3024
    Activity:
    Calpain inhibitor
    Chemical Name:
    Ac-Leu-Leu-Nle-CHO
    Alternate Names:
    Ac-LL-norleucinal
    Molecular Weight:
    383.53
    Molecular Formula:
    C20H37N3O4
    Solubility:
    Soluble in DMSO (up to 10 mg/ml) or in Ethanol (up to 5 mg/ml)
    Physical Properties:
    White solid
    Purity:
    98% by HPLC
    NMR (Conforms)
    Storage Temperature:
    -20°C
    Stability:
    Stable for 1 year from date of purchase as supplied. Solutions in DMSO or ethanol may be stored at -20°C for up to 1 month.
    Shipping Code:
    RT
    From $50.00
    View Product This product has multiple variants. The options may be chosen on the product page

  • Antipain 2HCl | Serine and cysteine protease inhibitor

    CAS:
    37682-72-7
    Catalog Number:
    10-2734
    Activity:
    Serine and cysteine protease inhibitor
    Chemical Name:
    (S)-1-Carboxy-2-phenylethyl]carbamoyl-L-arginyl-L-valyl-argininal, dihydrochloride
    Molecular Weight:
    677.62
    Molecular Formula:
    C27H44N10O6 • 2HCl
    Solubility:
    Soluble in Water (up to at least 10 mg/ml)
    Physical Properties:
    White solid
    Purity:
    98% by HPLC
    NMR (Conforms)
    Storage Temperature:
    -20°C
    Stability:
    Stable for 1 year from date of purchase as supplied. Solutions in distilled water may be stored at -20°C for up to 1 month.
    Shipping Code:
    RT
    From $35.00
    View Product This product has multiple variants. The options may be chosen on the product page

  • Belnacasan | ICE/caspase-1 inhibitor

    CAS:
    273404-37-8
    Catalog Number:
    10-4399
    Activity:
    ICE/caspase-1 inhibitor
    Chemical Names:
    (S)-1-((S)-2-(4-Amino-3-chlorobenzamido)-3,3-dimethylbutanoyl)-N-((2R,3S)-2-ethoxy-5-oxotetrahydrofuran-3-yl)pyrrolidine-2-carboxamide; VX-765
    Molecular Weight:
    508.99
    Molecular Formula:
    C24H33ClN4O6
    Solubility:
    Soluble in DMSO (>25 mg/ml)
    Physical Properties:
    Off-white to white solid
    Purity:
    98% HPLC
    NMR (Conforms)
    Storage Temperature:
    -20°C
    Stability:
    Stable for 1 year as supplied. Solutions in DMSO may be stored at -20°C for up to 3 months.
    Shipping Code:
    RT
    From $45.00
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  • Bestatin HCl | Aminopeptidase inhibitor

    CAS:
    65391-42-6
    Catalog Number:
    10-1286
    Activity:
    Aminopeptidase inhibitor
    Chemical Name:
    [(2S,3R)-3-Amino-2-hydroxy-4-phenylbutanoyl]-L-leucine HCl
    Molecular Weight:
    344.84
    Molecular Formula:
    C16H24N2O4 HCl
    Solubility:
    Soluble in Water (up to 10 mg/ml). Also soluble in DMSO and Ethanol.
    Physical Properties:
    White solid
    Purity:
    98% by TLC
    NMR (Conforms)
    Storage Temperature:
    -20°C (des.)
    Stability:
    Stable for 2 years from date of purchase as supplied. Solutions in DMSO, distilled water, or ethanol may be stored at -20° for up to 1 month.
    Shipping Code:
    RT
    From $40.00
    View Product This product has multiple variants. The options may be chosen on the product page

  • Chymostatin | Inhibitor of Chymotrypsin-like serine proteases

    CAS:
    9076-44-2
    Catalog Number:
    10-2722
    Activity:
    Inhibitor of chymotrypsin-like serine proteases
    Chemical Name:
    [(S)-1-Carboxy-2-phenylethyl]-carbamoyl-a-[2-amidohexahydro-4(S)-pyrimidyl]-(S)-glycyl-[A= Leu, B=Val, C=Ile]-phenylalaninal
    Molecular Weight:
    605.0 (ave.)
    Molecular Formula:
    C31H41N7O6
    Solubility:
    Soluble in DMSO (up to 20 mg/ml)
    Physical Properties:
    White or off-white solid
    Purity:
    96% by TLC
    NMR (Conforms)
    Storage Temperature:
    -20°C
    Stability:
    Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 1 month.
    Shipping Code:
    RT
    From $98.00
    View Product This product has multiple variants. The options may be chosen on the product page

  • DAPT | gamma-secretase inhibitor

    CAS:
    208255-80-5
    Catalog Number:
    10-4514
    Activity:
    γ-secretase inhibitor
    Alternate Names:
    LY-374973
    Chemical Name:
    N-[N-(3,5-Difluorophenacetyl)-L-alanyl]-S-phenylglycine t-butyl ester
    Molecular Weight:
    432.46
    Molecular Formula:
    C23H26F2N2O4
    Solubility:
    Soluble in DMSO (up to 18 mg/ml).
    Physical Properties:
    White solid
    Purity:
    98% by TLC
    NMR (Conforms)
    Storage Temperature:
    -20°
    Stability:
    Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20° for up to 3 months.
    Shipping Code:
    RT
    From $55.00
    View Product This product has multiple variants. The options may be chosen on the product page

  • E-64d | Cysteine protease inhibitor

    CAS:
    88321-09-9
    Catalog Number:
    10-1347
    Activity:
    Cysteine protease inhibitor
    Chemical Name:
    2S,3S-trans-(Ethoxycarbonyloxirane-2-carbonyl)-L-leucine-(3-methylbutyl)amide
    Molecular Weight:
    342.43
    Molecular Formula:
    C17H30N2O5
    Solubility:
    Soluble in DMSO (up to 20 mg/ml) or in Ethanol (up to 10 mg/ml).
    Physical Properties:
    White or off-white solid
    Purity:
    98% by HPLC
    NMR (Conforms)
    Storage Temperature:
    -20°C
    Stability:
    Stable for 1 year from date of purchase as supplied. Solutions in DMSO or ethanol may be stored at -20°C for up to 1 month.
    Shipping Code:
    RT
    From $40.00
    View Product This product has multiple variants. The options may be chosen on the product page

  • Elastatinal | Elastase inhibitor

    CAS:
    51798-45-9
    Catalog Number:
    10-2818
    Activity:
    Elastase inhibitor
    Chemical Name:
    N[(S)-1-Carboxyisopentyl]carbamoyl-a-[2-iminohexahydro-4(S)-pyrimidyl-(S)-glycl-(S)-glutaminyl-(S)-alaninal
    Molecular Weight:
    512.56
    Molecular Formula:
    C21H36N8O7
    Solubility:
    Soluble in DMSO (up to 3 mg/ml) or in Water (up to 5 mg/ml)
    Physical Properties:
    Lyophilized off-white solid
    Purity:
    98% by TLC
    NMR (Conforms)
    Storage Temperature:
    -20°C
    Stability:
    Stable for 1 year from date of purchase as supplied. Solutions in DMSO or distilled water may be stored at -20°C for up to 1 month.
    Shipping Code:
    RT
    From $75.00
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  • Ilomastat (GM-6001) | MMP inhibitor

    CAS:
    142880-36-2
    Catalog Number:
    10-1339
    Activity:
    MMP inhibitor
    Alternate Names:
    GM-6001
    Chemical Name:
    N-[(2R)-2-(Hydroxamidocarbonylmethyl)-4-methylpentanoyl]-L-tryptophan methylamide
    Molecular Weight:
    388.46
    Molecular Formula:
    C20H28N4O4
    Solubility:
    Soluble in DMSO (up to 10 mg/ml) or in Ethanol (up to 10 mg/ml).
    Physical Properties:
    White solid
    Purity:
    97% by TLC
    Storage Temperature:
    -20°
    Stability:
    Stable for 1 year from date of purchase as supplied. Solutions in DMSO or ethanol may be stored at -20° for up to 3 months.
    Shipping Code:
    RT
    From $52.00
    View Product This product has multiple variants. The options may be chosen on the product page

  • Leupeptin hemisulfate | Trypsin-like cysteine protease inhibitor

    CAS:
    103476-89-7
    Catalog Number:
    10-1346
    Activity:
    Trypsin-like cysteine protease inhibitor
    Alternate Names:
    Ac-Leu-Leu-Arg-CHO, hemisulfate
    Molecular Weight:
    475.59
    Molecular Formula:
    C20H38N6O4 &bul; 1/2H2SO4
    Solubility:
    Soluble in Water (up to 50 mg/ml). Also soluble in ethanol and methanol
    Physical Properties:
    White solid
    Purity:
    98% by HPLC
    NMR (Conforms)
    Storage Temperature:
    -20°C
    Stability:
    Stable for 1 year from date of purchase as supplied Solutions in distilled water, ethanol or methanol may be stored at -20°C for up to 3 months.
    Shipping Code:
    RT
    From $80.00
    View Product This product has multiple variants. The options may be chosen on the product page

  • MG-132 | Proteasome inhibitor

    CAS:
    133407-82-6
    Catalog Number:
    10-1309
    Activity:
    Proteasome inhibitor
    Alternate Names:
    Z-Leu-Leu-Leu-CHO
    Chemical Name:
    N-(Benzyloxycarbonyl)leucinylleucinylleucinal
    Molecular Weight:
    475.63
    Molecular Formula:
    C26H41N3O5
    Solubility:
    Soluble in DMSO (up to 45 mg/ml), in DMF (up to 45 mg/ml), or in Ethanol (up to 45 mg/ml).
    Physical Properties:
    White solid
    Purity:
    98% by HPLC
    Storage Temperature:
    -20°C
    Stability:
    Stable for 2 years from date of purchase as supplied. Solutions in DMSO, DMF or ethanol may be stored at -20° for up to 1 week.
    Shipping Code:
    RT
    From $50.00
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  • Nafamostat Mesylate | Serine protease inhibitor

    CAS:
    82956-11-4
    Catalog Number:
    10-1089
    Activity:
    Serine protease inhibitor
    Alternate Names:
    Futhan; FUT-175
    Chemical Name:
    6-Amidino-2-naphthyl-4-guanidinobenzoate dimesylate
    Molecular Weight:
    539.59
    Molecular Formula:
    C19H17N5O2·2CH4O3S
    Solubility:
    Soluble in Water (up to 25 mg/ml).
    Physical Properties:
    White solid
    Purity:
    98% by TLC
    NMR (Conforms)
    Storage Temperature:
    RT
    Stability:
    Stable for 2 years from date of purchase as supplied. Solutions in distilled water may be stored at 4°C for up to 1 month, or at -80°C for up to 6 months.
    Shipping Code:
    RT
    From $50.00
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  • P32/98 | DPPIV inhibitor

    CAS:
    136259-20-6
    Catalog Number:
    10-1142
    Activity:
    DPPIV inhibitor
    Alternate Names:
    Isoleucine thiazolidide hemi-fumarate
    Chemical Name:
    (2S,3S)-2-Amino-3-methyl-1-(thiazolidin-3-yl)pentan-1-one hemi-fumarate
    Molecular Weight:
    260.36
    Molecular Formula:
    C9H18N2OS·1/2(C4H4O4)
    Solubility:
    Soluble in DMSO (up to 25 mg/ml) or in Water (up to 20 mg/ml).
    Physical Properties:
    White solid
    Purity:
    98% by TLC
    NMR (Conforms)
    Storage Temperature:
    -20°C
    Stability:
    Stable for 2 years from date of purchase as supplied. Solutions in DMSO or distilled water may be stored at -20°C for up to 1 month.
    Shipping Code:
    RT
    From $100.00
    View Product This product has multiple variants. The options may be chosen on the product page

  • PD-150606 | Calpain Inhibitor

    CAS:
    179528-45-1
    Catalog Number:
    10-1515
    Activity:
    Calpain Inhibitor
    Chemical Name:
    (Z)-3-(4-Iodophenyl)-2-mercapto-2-propenoic acid
    Molecular Weight:
    306.12
    Molecular Formula:
    C9H7IO2S
    Solubility:
    Soluble in DMSO (up to 30 mg/ml) or in Ethanol (up to 15 mg/ml).
    Physical Properties:
    Yellow solid
    Purity:
    98% by TLC
    NMR (Conforms)
    Storage Temperature:
    -20°C (des.)
    Stability:
    Stable for 2 years from date of purchase as supplied. Solutions in DMSO or ethanol may be stored at -20° for up to 3 months.
    Shipping Code:
    RT
    From $69.00
    View Product This product has multiple variants. The options may be chosen on the product page

  • Pepstatin A | Aspartic protease inhibitor

    CAS:
    26305-03-3
    Catalog Number:
    10-1368
    Activity:
    Aspartic protease inhibitor
    Chemical Name:
    N-isovaleryl-L-valyl-L-valyl-3-hydroxy-6-methyl-γ-aminoheptanoyl-L-alanyl-3-hydroxy-6-methyl-γ-amino heptanoic acid
    Molecular Weight:
    685.90
    Molecular Formula:
    C34H63N5O9
    Solubility:
    Soluble in DMSO (up to 5 mg/ml) or in Ethanol (up to 1 mg/ml)
    Physical Properties:
    White solid
    Purity:
    98% by HPLC
    NMR (Conforms)
    Storage Temperature:
    -20°C
    Stability:
    Stable for 1 year from date of purchase as supplied. Solutions in DMSO or ethanol may be stored at -20°C for up to 2 months.
    Shipping Code:
    RT
    From $32.00
    View Product This product has multiple variants. The options may be chosen on the product page

  • Phosphoramidon | Neutral endopeptidase inhibitor

    CAS:
    119942-99-3
    Catalog Number:
    10-2548
    Activity:
    Neutral endopeptidase inhibitor
    Chemical Name:
    N-(α-Rhamnopyranosyloxyhydroxyphosphinyl)-L-leucyl-L-tryptophan•2Na
    Molecular Weight:
    587.47
    Molecular Formula:
    C23H32N3O10P • 2Na
    Solubility:
    Soluble in DMSO, methanol, or distilled water
    Physical Properties:
    White solid
    Purity:
    97% by TLC
    NMR (Conforms)
    Storage Temperature:
    -20°C
    Stability:
    Stable for 2 years from date of purchase as supplied. Solutions in DMSO, methanol, or distilled water may be stored at -20°C for up to 2 months.
    Shipping Code:
    RT
    From $100.00
    View Product This product has multiple variants. The options may be chosen on the product page

  • Talabostat mesylate | Pyroptosis inducer / Inflammasome activator

    CAS:
    150080-09-4
    Catalog Number:
    10-4005
    Activity:
    Pyroptosis inducer / Inflammasome activator
    Chemical Name:
    ((2R)-1-((2S)-2-Amino-3-methylbutanoyl)pyrrolidin-2-yl)boronic acid methanesulfonate
    Alternate Names:
    Val-boroPro; PT-100
    Molecular Weight:
    310.18
    Molecular Formula:
    C9H19BN2O3 • CH3SO3H
    Solubility:
    Soluble in DMSO (up to at least 25 mg/ml)
    Physical Properties:
    White solid
    Purity:
    97% by HPLC
    NMR (Conforms)
    Storage Temperature:
    -20°C
    Stability:
    Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 1 month.
    Shipping Code:
    RT
    From $60.00
    View Product This product has multiple variants. The options may be chosen on the product page

  • TPCK | Serine protease inhibitor

    CAS:
    402-71-1
    Catalog Number:
    10-2290
    Activity:
    Serine protease inhibitor
    Chemical Name:
    N-p-Tosyl-L-phenylalanine chloromethyl ketone
    Molecular Weight:
    351.8
    Molecular Formula:
    C17H18ClNO3S
    Solubility:
    Soluble in DMSO (up to 10 mg/ml).
    Physical Properties:
    White solid
    Purity:
    98% by TLC
    NMR (Conforms)
    Storage Temperature:
    -20°
    Stability:
    Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20° for up to 3 months.
    Shipping Code:
    RT
    From $32.00
    View Product This product has multiple variants. The options may be chosen on the product page

  • Z-DEVD-FMK | Caspase-3 inhibitor

    CAS:
    210344-95-9
    Catalog Number:
    10-2904
    Activity:
    Caspase-3 inhibitor
    Chemical Names:
    Benzyloxycarbonyl-Asp(OMe)-Glu(OMe)-Val-Asp(OMe)-fluoromethylketone
    Molecular Weight:
    668.67
    Molecular Formula:
    C30H41FN4O12
    Solubility:
    Soluble in DMSO (20 mg/ml)
    Physical Properties:
    Lyophilized solid
    Purity:
    >98% TLC
    NMR (Conforms)
    Storage Temperature:
    -20°C
    Stability:
    Stable for 2 years from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 1 month.
    Shipping Code:
    RT
    $110.00
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  • 10-4990 ZLeuLeuLeuVS chemical structure

    Z-Leu-Leu-Leu-vinylsulfone | Proteasome inhibitor

    CAS:
    193482-47-2
    Catalog Number:
    10-4990
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  • Z-VAD-FMK | Caspase inhibitor

    CAS:
    187389-52-2
    Catalog Number:
    10-2614
    Activity:
    Caspase inhibitor
    Alternate Names:
    ZVAD(OMe)-FMK
    Chemical Name:
    Benzyloxycarbonyl-Val-Ala-Asp(OMe)-fluoromethylketone
    Molecular Weight:
    467.5
    Molecular Formula:
    C22H30FN3O7
    Solubility:
    Soluble in DMSO (up to 10 mg/ml).
    Physical Properties:
    Lyophilized or waxy solid
    Purity:
    98% by TLC
    NMR (Conforms)
    Storage Temperature:
    -20°C
    Stability:
    Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20° for up to 1 week.
    Shipping Code:
    RT
    $98.00
    View Product This product has multiple variants. The options may be chosen on the product page

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